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5-{[2-(diethylamino)ethyl](methyl)amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 1-benzyl-3-cyclopropaneamido-5-[(1-hydroxypropan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(benzylsulfamoyl)(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)amine
1-(4-chlorophenyl)-4-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-5-methylpiperazin-2-one
1-ethyl-N-(1H-imidazol-2-ylmethyl)-N-methyl-1H-indole-5-carboxamide
(2S)-2-amino-N-[(2-methylphenyl)methyl]-3-phenyl-N-(prop-2-en-1-yl)propanamide
N-[2-(dimethylamino)ethyl]-N-methyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}cyclohexanecarboxamide
(3R,4R)-4-amino-1-[4-(4-methylphenoxymethyl)benzoyl]piperidin-3-ol
N-[3-(2-ethoxyphenyl)propyl]-2,6-dimethylpyridine-4-carboxamide
N-(1-{2-[4-(3-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-4-oxo-4-phenylbutanamide
2-(3-methoxypropyl)-9-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[1-(1-methylazepane-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-(4-fluorophenyl)-4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazine
methyl 5-[2-(morpholin-4-yl)butanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[(2-chloro-6-fluorophenyl)methyl]-N,2-diethylpyrimidine-5-carboxamide
methyl 4-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}-4-oxobutanoate
5-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-(1H-inden-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-fluoro-4-[(3R,4R)-3-hydroxy-4-(morpholin-4-yl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
3-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-N-(1-methyl-1H-imidazol-2-yl)benzamide
N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-[2-(phenylsulfanyl)ethyl]acetamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-3-yl]methanol
4,4-difluoro-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperidine
N,4-diethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-1,3-thiazole-5-carboxamide
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
3-ethyl-1-[3-(3-methoxyphenyl)phenyl]-3-[(1-methylpyrrolidin-3-yl)methyl]urea
methyl[(4-methyl-1H-imidazol-2-yl)methyl][(3-phenyl-1H-pyrazol-5-yl)methyl]amine
2-{1-[(3,4-difluorophenyl)methyl]-4-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N,2,6-trimethyl-4-oxo-N-[(4-phenoxyphenyl)methyl]-1,4-dihydropyridine-3-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
5-cyclopropanecarbonyl-1'-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-6-(pyrrolidin-1-yl)pyrimidine
methyl (2S)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidine-2-carboxylate
1-(carbamoylmethyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidine-3-carboxamide
1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}azocane
4-ethyl-3-{2-[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
9-[(4-acetylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)propanamide
2-[(2-chlorophenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}morpholine
2-({[(3R,4R)-4-(hydroxymethyl)-1-[3-(trifluoromethyl)benzoyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-(dimethylamino)-N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)-2-(3-methylphenyl)acetamide
N-[4-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)phenyl]acetamide
8-(1-methyl-1H-pyrazole-5-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
5-methyl-1-{4-[(prop-2-en-1-yl)carbamoyl]phenyl}-1H-pyrazole-3-carboxylic acid
(4aS,7aR)-1-(1,2-oxazole-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
(1R,7S)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-3-[2-(pyridin-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one