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N-{1-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methylphenol
(benzylsulfamoyl)[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amine
8-(5-chloropyridin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
N-({1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-2,2-dimethylpropanamide
3-cyclobutyl-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
7-[(2-chloro-6-fluorophenyl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
3-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1-[4-(propylsulfanyl)phenyl]urea
N-(3-hydroxy-2,2-dimethylpropyl)-5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
(3S,4R)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2,5-dimethoxybenzene-1-sulfonamide
N-cyclopropyl-2-{methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}pyridine-4-carboxamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-(3-chlorophenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
methyl 2-(N-methyl-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)acetate
N-(2-methoxyethyl)-2-(1-methyl-1H-imidazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
8-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(carbamoylmethyl)-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)piperidine-3-carboxamide
4-(cyclopropylmethyl)-1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(2-methylpropanoyl)piperidine-2-carboxamide
4-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-(oxolane-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-fluoro-N-[4-(4-{[1-(thiophen-2-yl)propyl]amino}piperidin-1-yl)phenyl]benzamide
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}pent-4-enamide
2-methyl-6-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}phenol
4-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrimidin-2-amine
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(4aS,7aR)-1-(4-methylpyridine-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclohexyl-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(4-methylpyridin-2-yl)propyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2,5-difluorobenzamide
3-({8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)benzonitrile
2-cyclopropyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,3-benzoxazole-6-carboxamide
(2S,4R)-4-amino-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-N-methylpyrrolidine-2-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
N-(3-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}pyridin-2-yl)-2,2-dimethylpropanamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}propanamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
5-methyl-4-{[2-(methylsulfamoyl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxylic acid
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
6-{2-oxa-7-azaspiro[4.5]decan-7-yl}-9H-purin-2-amine
1-(5-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)pyrrolidine
3-(dimethyl-1H-1,2,4-triazol-1-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,2-dimethylpropanamide
5-fluoro-N-methyl-2-(2,4,6-trimethylphenyl)pyrimidin-4-amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]propanamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
[(1-ethyl-1H-pyrazol-4-yl)methyl](methyl)[2-(pyridin-2-yl)ethyl]amine