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3-(aminomethyl)-4-[(2-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
2-(3,4-dichlorophenyl)-4-(3-ethyl-1,2-oxazole-5-carbonyl)morpholine
3-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-3,4-dihydro-2H-1λ6,2-benzothiazine-1,1-dione
1-(3-{2-methyl-2,7-diazaspiro[4.5]decane-7-carbonyl}phenyl)imidazolidin-2-one
3-{2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}cyclohex-3-ene-1-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
3-{[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-(2-fluoroethyl)benzamide
1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
N-cyclopropyl-1-{2-[1-(3-methylbenzoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[2-methoxy-4-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(2-fluorophenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-3-[(methylsulfanyl)methyl]piperidine
(2R,6R)-4-{[(furan-2-ylmethyl)carbamoyl]methyl}-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
7-fluoro-3-{[4-methoxy-4-(prop-2-en-1-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
5-chloro-2-[3-(3-methoxypropyl)piperidine-1-carbonyl]phenol
[(3R,4R)-1-(5-methyl-1H-indazole-3-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(3-fluorophenyl)-N-(2-{octahydropyrrolo[1,2-a]piperazin-2-yl}-2-oxoethyl)methanesulfonamide
1-({1-[(3-methoxyphenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}methyl)-4-phenylpyrrolidin-2-one
5-(4-methyl-3-phenylpiperazine-1-carbonyl)-4-(trifluoromethyl)pyrimidin-2-amine
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
(3S,7S)-5-(1-ethyl-1H-pyrazole-5-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-methoxypropanamide
3-({3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}methyl)-6,8-dimethyl-1,2-dihydroquinolin-2-one
1-{2-[2-(3-phenylpropyl)morpholine-4-carbonyl]phenyl}ethan-1-one
8-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-N-(cyclopropylmethyl)-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(3-hydroxyphenyl)-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}ethan-1-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-[(3-fluorophenyl)methyl]-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-[3-(cyclopentyloxy)propyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
4-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-ethylpiperidine
N-(2H-1,3-benzodioxol-5-yl)-3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanamide
4-(2-methylquinazolin-4-yl)benzamide
3-fluoro-4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-(6-methoxynaphthalen-2-yl)-4-[2-(1H-pyrazol-1-yl)ethyl]morpholine
3-methoxy-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidine
5-(2-methoxyphenyl)-3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)azepane
2-(3,4-dimethoxyphenyl)-3-[(4-methoxypiperidin-1-yl)methyl]-7-methylquinoline
N-({1-[(4,5-dimethylthiophen-2-yl)methyl]pyrrolidin-3-yl}methyl)-2-acetamidoacetamide
4-acetyl-N-[3-(2-methylpyrimidin-4-yl)phenyl]-1,4-diazepane-1-carboxamide
3,5-dimethyl-2-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1,4-dihydropyridin-4-one
N-methyl-5-{[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-2-(3,4,5-trimethoxyphenyl)pyridine
methyl 5-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(2S,4R)-N-ethyl-4-(4-{[1-(5-fluoro-2-methylphenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide