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2-[(3R,4S)-3-acetamido-4-propylpyrrolidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(dimethylamino)benzamide
3-[2-(azepan-1-yl)-2-oxoethyl]-1-[2-(dimethylamino)ethyl]-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
3-({4-[3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
6-methyl-N-propyl-5-[5-(pyridin-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
7-(2-methoxyethyl)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1,5-dimethyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
4-(cyclopropylmethyl)-1-[(4-hydroxy-2,6-dimethylphenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
(1R,5R)-6-(2-methoxyethyl)-3-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-{4-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]phenyl}acetamide
N-[(1-methylpiperidin-3-yl)methyl]-2-propoxybenzamide
N-[(3-methoxyphenyl)methyl]-2-methyl-N-propyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl][(2,5-dimethylfuran-3-yl)methyl]methylamine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(propan-2-yl)-6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-amine
3-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]phenol
(1S,5R)-3-[(3-chloro-4-methoxyphenyl)methyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-[({1,9-dioxaspiro[5.5]undecan-4-yl}amino)methyl]-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
methyl 2-(7-chloro-3-{[4-(hydroxydiphenylmethyl)piperidin-1-yl]methyl}-2-oxo-1,2-dihydroquinolin-1-yl)acetate
5-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}-2-methoxybenzoic acid
N-[3-(furan-2-yl)phenyl]-1-[2-(thiophen-3-yl)acetyl]piperidine-4-carboxamide
4-(methylamino)-N-{[1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]methyl}benzamide
5-fluoro-2-(1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)cyclopropanamine
{[7-fluoro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}[1-(thiophen-2-yl)ethyl]amine
methyl (3S)-2-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-3-carboxylate
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(1H-pyrrol-1-yl)propanamide
N-(2-methoxyethyl)-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-{4-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)thiomorpholine-4-carboxamide
N-butyl-N-methyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
1-(4-chlorophenyl)-4-(2-fluoro-6-methoxybenzoyl)-5-methylpiperazin-2-one
5-fluoro-3-methyl-2-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1H-indole
N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-hydroxy-1-(2-methoxyethyl)-3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]piperidin-2-one
3-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
6-methoxy-3-[4-(morpholin-4-yl)piperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
9-(2-fluorobenzoyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
[(3-ethoxy-4-methoxyphenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
2-ethyl-1-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-2,5-dihydro-1H-pyrrole
4-[1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperidin-4-yl]thiomorpholine
(4S)-1-[(5-fluoro-2-methoxyphenyl)methyl]-3,3,4-trimethylpiperidin-4-ol
2-(1H-imidazol-2-yl)-N-[(8-methoxyquinolin-5-yl)methyl]-N-methylbenzamide
1-(3,5-dimethylphenyl)-4-(4-methylpyrimidin-2-yl)piperazin-2-one
5-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-3-yl)imidazolidine-2,4-dione