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1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
7-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
4-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
6-ethyl-4-{[(3R)-3-fluoropyrrolidin-1-yl]methyl}-2H-chromen-2-one
3-[2-(4-fluorophenyl)acetyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[1-(2-cyclohexylacetyl)piperidin-3-yl]methyl}-4-fluorobenzamide
6-phenyl-N-[(1R,2S)-2-phenylcyclopropyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(methoxymethyl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}cyclobutane-1-carboxamide
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
1-{3-[3-(4-tert-butylbenzoyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
4-ethyl-3-[(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(3-methylphenyl)phenyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-3-carboxamide
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-{4-methyl-6-[(1H-1,2,3,4-tetrazol-5-ylmethyl)amino]pyrimidin-2-yl}phenol
3-methyl-3-phenyl-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]butan-1-one
7-(3-methoxypropyl)-2-(quinolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{3-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
3-methyl-5-(4-methyl-1H-imidazol-5-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
3-[(2-fluorophenyl)formamido]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)[2-(piperidin-1-yl)ethyl]amine
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-[(2,3-dichlorophenyl)methyl]-4-methylazepan-4-ol
N-methyl-4-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
2-methoxy-1-[1'-(1-methylpiperidine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-cyclopropyl-N-ethyl-4-hydroxy-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]pyrimidine-5-carboxamide
1-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}azepan-2-one
4-[(2-amino-5,6-dimethylpyrimidin-4-yl)amino]-1-(3-chlorophenyl)pyrrolidin-2-one
N,N-diethyl-5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]propanamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-1,2,3-triazole
[(dimethyl-1,2-oxazol-4-yl)methyl][(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]methylamine
(4aS,7aR)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-(2,6-dimethoxybenzoyl)-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
methyl[(3-methylpyridin-4-yl)methyl]{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
2-(4-fluorophenyl)-2-hydroxy-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(4,6-dimethylpyridin-2-yl)benzamide
1-(1-benzoxepine-4-carbonyl)-4-hydroxypiperidine-4-carboxylic acid
2-(2,3-dimethylphenoxy)-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]acetamide
4-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-N,N-dimethyl-4-oxobutanamide
N-(1-benzylpiperidin-4-yl)-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]acetamide
{2-[6-(benzyloxy)pyridin-3-yl]pyridin-4-yl}methanol
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[2-(piperidin-1-yl)ethyl]benzamide
1-{6-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridin-3-yl}ethan-1-one
ethyl({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine