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methyl (2R,4S)-4-hydroxy-1-({2-oxo-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-4-yl}methyl)piperidine-2-carboxylate
N-(2-{1-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]piperidin-2-yl}ethyl)acetamide
N-cyclobutyl-4-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]sulfonyl}benzamide
3-(2-methoxyphenoxy)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}azetidine
N-[(2S)-1-oxo-1-(3-oxo-4-phenylpiperazin-1-yl)propan-2-yl]acetamide
3-[2-methyl-2-(morpholin-4-yl)propyl]-3,9-diazaspiro[5.5]undecane
2-(1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
(3aR,6aS)-5-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(1H-pyrrol-1-yl)ethyl]amino}methyl)piperidin-2-one
1-(2-methylpropyl)-4-oxo-N-[(4-phenyloxan-4-yl)methyl]-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-3-(1-methylpiperidin-2-yl)propan-1-one
N,8-dimethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[(2,6-difluorophenyl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(2-hydroxyethyl)pyrrolidin-3-yl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
(1S,4S)-2-(2H-1,3-benzodioxol-5-yl)-5-{[4-(trifluoromethoxy)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[(1,2-oxazol-3-ylmethyl)amino]methyl}piperidin-2-one
3-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]-1-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}urea
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-{1-oxaspiro[4.4]nonan-3-yl}urea
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}amino)pyridine-3-carboxamide
2-{4-[(2-fluorophenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-(3,4,5-trimethoxyphenyl)ethan-1-one
1-(carbamoylmethyl)-N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]piperidine-4-carboxamide
1-{7-[2-hydroxy-4-(1H-pyrazol-1-yl)butan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-3-phenylprop-2-yn-1-one
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
(3S,4R)-1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
1-cyclopentyl-3-(4-methoxyphenyl)-3-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione
(2R,3R)-1'-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N3-[(3-fluoro-4-methylphenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(6-methyl-2-propylpyrimidin-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-amine
(4aS,8aR)-6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
2,4-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidine-5-carboxamide
4-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}azetidin-3-yl)morpholine
2-[4-(2-methoxybenzenesulfonamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
(butan-2-yl)[(4-methanesulfonylphenyl)methyl](3-phenylprop-2-yn-1-yl)amine
2-(4-fluoro-2-methylphenyl)-N-[1-(2-methoxyphenyl)ethyl]-N-methylacetamide
methyl (2R,4S)-1-[(1-ethyl-1H-indol-6-yl)methyl]-4-hydroxypiperidine-2-carboxylate
(2S,4S)-1-benzyl-N-ethyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
1-{1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperidin-4-yl}piperidin-4-ol
({4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-(furan-3-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-fluorobenzene-1-sulfonamide
ethyl 4-{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine-1-carboxylate
1-[4-(ethylsulfanyl)phenyl]-3-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]urea
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-ethoxypropan-1-one
3-methoxy-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine
9-(5,6-dimethoxypyrazine-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-[4-(dipropylamino)piperidin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
4-[4-(morpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]-N-[(1S)-1-phenylethyl]piperidine-1-carboxamide