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1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[(1-hydroxycyclohexyl)methyl]amino}methyl)piperidin-2-one
1-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
3-(4-fluorophenyl)-N-methyl-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
1-{3-[2-(3-methoxyphenyl)pyrrolidin-1-yl]propyl}-5-methyl-1H-1,2,3,4-tetrazole
2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidin-4-ol
1-(3-benzyl-1H-1,2,4-triazol-5-yl)naphthalen-2-ol
2-[2-(1H-imidazol-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-(piperidine-1-carbonyl)benzene-1-sulfonamide
N-(1-cycloheptylpiperidin-3-yl)-4-methyl-1,3-oxazole-5-carboxamide
2-methoxy-1-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)ethan-1-one
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-(2-methoxyethyl)-4-oxo-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N,3-dimethyl-N-(oxolan-3-yl)-5-propyl-1-benzofuran-2-carboxamide
2-methoxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
2-{2-[2-(2-hydroxyethyl)morpholin-4-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-[(propan-2-yl)amino]pyridine-3-carboxamide
6-(8-methoxy-2-methylquinolin-5-yl)-N-methylpyridine-2-carboxamide
1-(4-ethylpiperazin-1-yl)-3-(1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)propan-1-one
1-methyl-2-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
1-(ethanesulfonyl)-3-(3-fluoro-4-phenylbenzoyl)piperidine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-chloropyridin-2-yl)piperidin-3-ol
(3S,9aR)-3-benzyl-8-(3-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(3-{3-[4-(pyrrolidin-1-ylmethyl)phenyl]phenyl}-1H-pyrazol-1-yl)propan-1-ol
4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)-N-(2-methyl-1-benzofuran-7-yl)piperazine-1-carboxamide
N3-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-4-oxo-N5-[2-(propan-2-yloxy)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(1,2-benzoxazol-3-yl)-1-[3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
methyl 5-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-{4-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
3-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]piperidin-2-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-1H-pyrazole-3-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2,4-dimethoxybenzamide
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-methoxy-N-[2-(propane-2-sulfonyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[3-(4-{[1-(2-methylpropyl)cyclopropyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(6-methylpyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
1-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-{1-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperidin-3-yl}ethan-1-amine
2-acetamido-3-methyl-N-({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)butanamide
8-(4-oxo-4-phenylbutyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[4-({[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}methyl)phenyl]butanamide
6-(2-aminoethyl)-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,2-dimethylpyrimidin-4-amine
N-(3-phenylpropyl)-6-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-[3-(dimethylcarbamoyl)-5-({[(2-ethoxyphenyl)methyl]amino}methyl)phenyl]pyridine-2-carboxamide
2-ethyl-4-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine