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5-cyclopropanecarbonyl-1'-{[2-(methylsulfanyl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-[5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,3-benzodiazole
3-[4-(dimethylamino)phenyl]-1-[4-(1-methylpiperidin-4-yl)piperazin-1-yl]propan-1-one
2-[(3,5-difluorophenyl)methyl]-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-methoxyethoxy)acetamide
1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[4-(azepan-1-yl)butyl]-6-(methoxymethyl)pyrimidin-4-amine
N-[(3S,5S)-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrrole-2-carboxamide
N5-butyl-N3-(cyclopropylmethyl)-1-(furan-2-ylmethyl)-4-oxo-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
2-(2-methyl-1,3-thiazol-4-yl)-N-[(3-methyl-1-benzofuran-2-yl)methyl]acetamide
ethyl 4-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]piperidine-1-carboxylate
3,5-difluoro-2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
2-[4-(benzyloxy)-2-fluorophenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
(3S,4R)-1-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-cyclopentyl-N5-[(3-fluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(1H-imidazol-1-yl)butan-2-yl]acetamide
2-ethyl-8-[2-(4-ethylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-methoxyethyl (4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
methyl 2-(morpholine-4-sulfonyl)-6-[(2,4,5-trimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
{5-fluoro-7-[5-(methanesulfonylmethyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}cyclobutane-1-carboxamide
5-{[(3-chlorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine
1-ethyl-N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-2-carboxamide
4-[4-(furan-2-yl)benzoyl]-7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4R)-4-{[(4-chlorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
2-[9-(3-hydroxy-4-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
3-{[(1-benzylpyrrolidin-3-yl)amino]methyl}-6-chloro-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine-4-carboxylic acid
N-benzyl-2-(2,5-dioxoimidazolidin-1-yl)-N-[(4-methyl-1,3-thiazol-5-yl)methyl]acetamide
4-[(5-ethylfuran-2-yl)methyl]-2-[(4-methoxyphenyl)methyl]morpholine
1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}azetidin-3-ol
3-(cyclohex-1-en-1-ylmethyl)-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
(2E)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(pyridin-3-yl)prop-2-enamide
N-[2-(1-{2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetyl}piperidin-2-yl)ethyl]acetamide
8-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-(oxolan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
2-({[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
1-cyclohexanecarbonyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrrolidine-2-carboxamide
(3S,4S)-1-(cyclohexylcarbamoyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
N-({7-[3-(4-fluorophenyl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-(2-phenoxyethyl)-4-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperazine
4-(4-butylpiperazine-1-carbonyl)-1,2-dihydroquinazolin-2-one
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one