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{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
1-[1-(4-methoxyphenyl)-2,2-dimethylcyclopropanecarbonyl]-4-(pyridin-4-yl)piperazine
2-(4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
1-{4-[(3-hydroxypropyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-[1-(4-methanesulfonylphenyl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-3-carboxamide
1-(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)-2-(thiophen-2-yl)ethan-1-one
N-(4-fluoro-2-methylphenyl)-3-{1-[2-(pyridin-2-ylsulfanyl)acetyl]piperidin-3-yl}propanamide
(1S,5R)-3-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-ethylpentan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)piperazin-2-one
1-(5-chloropyridin-2-yl)-4-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperazine
4-{4-[(2-ethoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-(2-{1-[3-(3,4-dimethoxyphenyl)propanoyl]piperidin-2-yl}ethyl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-(oxolan-3-yl)-4-(thiomorpholine-4-sulfonyl)benzamide
5-methoxy-2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyrimidine
3-benzyl-1-methyl-3-[3-oxo-3-(pyrrolidin-1-yl)propyl]-2,3-dihydro-1H-indol-2-one
phenyl (7R,9aR)-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-(oxolan-2-ylmethyl)-1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
6-methyl-2-[3-({methyl[2-(morpholin-4-yl)ethyl]amino}methyl)phenyl]-5-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidine-4-carbonitrile
(3S)-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
4-chlorophenyl (7R,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2,3,6-trimethylquinoline-4-carboxamide
4-ethoxy-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine
4-[(3-methylphenyl)sulfanyl]-N-(1-propyl-1H-1,2,3-triazol-4-yl)piperidine-1-carboxamide
3-ethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
1-[1-(4-cyanobenzoyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
8-(1,3-benzothiazol-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(quinolin-4-ylmethyl)-1,4-diazepan-5-one
3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]pyridin-2-amine
ethyl 1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxylate
4-[(4-chloro-3-fluorophenyl)methyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
2-oxo-1-phenyl-N-[3-(propan-2-yloxy)propyl]pyrrolidine-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-1,3-oxazole-5-carboxamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)propanamide
4-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-4-(4-methylpiperazin-1-yl)benzamide
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
3,5,7-trimethyl-2-[4-(2-methylpyridin-4-yl)piperazine-1-carbonyl]-1H-indole
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-methyl-4-phenylpiperazine
2-ethyl-8-(3-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-fluoro-1,3-dimethyl-2-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-indole
2-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}-6-ethoxyphenol
(2R,3R,6R)-5-[(2,4-difluorophenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane