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1-(benzenesulfonyl)-N-(3,4-dimethoxyphenyl)piperidin-3-amine
ethyl 5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2-phenylethyl)-6-[(2E)-3-phenylprop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
methyl (2S)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
3-benzyl-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{imidazo[1,2-a]pyridin-3-yl}-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
N-[2-(3-chlorophenyl)ethyl]-3-[5-(5-methyl-1,2-oxazol-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-(1-{7-[(4-chlorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
2-(4-fluorophenyl)-N-[2-(7-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
methyl 3-ethyl-2-[3-(1H-pyrazol-3-yl)phenyl]-3H-imidazo[4,5-b]pyridine-6-carboxylate
3-[2-(3-fluorophenyl)azepane-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
2-(thiophen-3-ylmethyl)-4-{4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-methoxy-2-({4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-[2-(dimethylsulfamoyl)ethyl]-2-fluoro-5-sulfamoylbenzamide
(2E)-1-{4-[2-(4-methylphenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-(thiophen-2-yl)prop-2-en-1-one
4-[(2,3-dichlorophenyl)methyl]-2-(2-methoxyethyl)morpholine
3,3-bis(2-methoxyethyl)-1-[3-(4-methylpiperazine-1-carbonyl)phenyl]urea
2-methoxy-1-{4-[(8-methoxy-2H-chromen-3-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
2-methyl-3-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}phenol
2-({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
2-[4-(1H-imidazol-1-yl)butanoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-({[(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amino}methyl)-4H-chromen-4-one
1-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-methylbut-2-en-1-one
1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-methyl-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-fluoropyrimidin-2-amine
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
(2E)-3-(2-chlorophenyl)-N-(oxolan-2-ylmethyl)-N-{[4-(pyridin-3-ylmethoxy)phenyl]methyl}prop-2-enamide
1-(difluoromethyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H-pyrazole-3-carboxamide
4-[5-(2,3-dihydro-1-benzofuran-7-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]-3,5-dimethyl-1,2-oxazole
N-[(4-cyanophenyl)methyl]-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-(5-acetylthiophen-3-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl (2S,4R)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-[(2,5-dimethylphenyl)methyl]pyrrolidine-2-carboxylate
N,N-dimethyl-3-[2-({[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]carbamoyl}amino)phenyl]propanamide
1,4-dimethyl-9-[6-(propan-2-yl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.5]undecane
3-[2-(dimethylamino)ethyl]-5-[1-(furan-3-ylmethyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
4-chloro-1-methyl-3-({4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)-1H-indazole
3-(4-chloro-1H-pyrazol-1-yl)-1-(6-hydroxy-1,4-oxazepan-4-yl)propan-1-one
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(oxolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[(1R,3S)-3-(cyclobutylcarbamoyl)cyclopentyl]-5-methyl-1-[(methylcarbamoyl)methyl]-1H-pyrazole-3-carboxamide
2-[4-(3-fluoropyridin-4-yl)piperazin-1-yl]-1,3-benzothiazole
5-(4-chloro-2-methoxyphenoxymethyl)-N-[(3,4-difluorophenyl)methyl]-1,2-oxazole-3-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(morpholin-4-yl)benzamide
N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(oxan-4-yl)pyrrolidin-3-amine
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-indazole