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6-[(3-methoxyphenyl)methoxy]-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(2-phenylethyl)-1,4-diazepan-2-one
2-phenoxy-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
3-{[(4-fluoro-3-methoxyphenyl)methyl]amino}-5-(4-methyl-1,4-diazepane-1-carbonyl)-N-phenylbenzene-1-sulfonamide
1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-[(dimethylamino)methyl]azepan-4-ol
N-phenyl-5-[2-(phenylformamido)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)ethan-1-one
N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
N4-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-amino-N-cyclopropyl-3-ethyl-N-(1H-indol-5-ylmethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-amino-2-methyl-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
2-(methoxymethyl)-6-methyl-N-[3-(morpholin-4-yl)propyl]-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
(3aS,6aR)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazole
{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(1H-pyrazol-1-yl)phenyl]methyl}amine
1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyrrolidin-1-yl)propan-1-one
3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-[4-(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-2-phenylethan-1-one
(5-{1-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
N,4-dimethyl-2-phenyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
2-(2-hydroxyphenoxy)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
1-(2-aminoethyl)-N-{[4-(butan-2-yloxy)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{2-oxo-4-[2-(propylsulfanyl)pyrimidin-5-yl]-1,2,3,4-tetrahydroquinolin-7-yl}acetamide
(1S,5R)-6-(3-fluoro-4-methoxybenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[4-(2-hydroxypyridin-3-yl)phenyl]acetamide
4-[(2,3-dimethoxyphenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
3-[4-(ethoxycarbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carbonyl]pyridin-1-ium-1-olate
4-(4-{[4-(9H-purin-6-yl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(4-phenyloxan-4-yl)methyl]furan-2-carboxamide
1-[5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-(1-benzothiophen-2-ylmethyl)-1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-butyl-3-({[2-(4-fluorophenyl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(4-{[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}-6-methylpyrimidin-2-yl)phenol
(3S,4R)-4-(3-fluorophenyl)-1-(1-methyl-1H-indole-4-carbonyl)pyrrolidine-3-carboxylic acid
6-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
4-(4-chlorophenoxy)-N-(oxan-2-ylmethyl)piperidine-4-carboxamide
7-(cyclopropylmethyl)-2-[4-(methylsulfanyl)benzoyl]-2,7-diazaspiro[4.5]decane
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-2,3,6-trimethylquinoline
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethan-1-one
ethyl (4aS,8aR)-6-[2-(methylsulfanyl)pyrimidin-4-yl]-decahydro-1,6-naphthyridine-4a-carboxylate
{3-benzyl-1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}methanol
N-(2-{[3-(1H-imidazol-2-yl)phenyl]formamido}ethyl)propanamide
N-[4-chloro-3-(dimethylcarbamoyl)phenyl]-3-propoxypiperidine-1-carboxamide
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
1-(3-methyl-3-phenylpiperidin-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one