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2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
6-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[1'-(2-hydroxy-4-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-[3-(furan-2-yl)phenyl]-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxamide
5-chloro-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
(3S,4S)-3-hydroxy-4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-1λ6-thiolane-1,1-dione
N-(2-hydroxyethyl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(propan-2-yl)benzamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxyethan-1-one
2-[2-({[(3S)-1-benzylpyrrolidin-3-yl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
2-(1-cyclopentyl-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
2-(3-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)ethan-1-ol
1-benzyl-4-(2-phenylethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-(2-phenylethyl)acetamide
3-{[(1-methoxypropan-2-yl)amino]methyl}-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-(3-cyclopropylpropanoyl)-N-(oxolan-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-3-carboxamide
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)thiophene-2-carboxamide
4-{3-[(4-cyclopentylpiperazin-1-yl)methyl]-8-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine
[(2,3-dimethoxyphenyl)methyl]({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
N-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}-N-cyclopropyl-2-methylpropanamide
5-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
(3S)-3-ethyl-4-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]morpholine
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
[(4-{[6-(2-methoxyphenyl)pyridazin-3-yl]oxy}phenyl)methyl]dimethylamine
5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3,5-dimethyl-2-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-indole
N3-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
1-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-ethylpiperidine-3-carboxylic acid
4-(3-chloro-4-fluorobenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(1S,5R)-6-(3-chlorobenzoyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(4,4-difluoropiperidin-1-yl)-N-ethylpyrimidin-4-amine
N'-cyclopentyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}butanediamide
N-methyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1R,5S)-6-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)-6-azabicyclo[3.2.1]octane
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
(2S,4R)-4-amino-1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(5-methylpyrimidin-2-yl)-1-oxa-8-azaspiro[4.5]decan-3-amine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-(3-methoxyphenyl)azetidin-1-yl]propan-1-one
(2S)-2-amino-1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-phenylethan-1-one
4-{5-[(cyclopentylamino)methyl]-2-methoxyphenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
(2S,4R)-4-amino-1-(4-chloro-3-fluorobenzoyl)-N,N-diethylpyrrolidine-2-carboxamide
3-(ethoxymethyl)-1-methyl-5-[2-(methylsulfanyl)-1,3-thiazol-4-yl]-1H-1,2,4-triazole
3-amino-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidine-3-carboxylic acid
N-{3-[2-(2-ethylpyrimidin-5-yl)-1H-imidazol-1-yl]phenyl}pyridine-3-carboxamide
2-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)-6-methoxyphenol
2-methyl-6-[3-(2-phenylethyl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one