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5-[4-(1,3-benzoxazol-2-yl)piperidine-1-carbonyl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl]({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(4-methylpiperidin-1-yl)acetamide
2-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}phenol
3-methyl-1-(2-methyl-1-benzofuran-5-yl)-3-[(1-phenylpyrrolidin-3-yl)methyl]urea
5-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-ethyl-1,2,4-oxadiazole
2,6-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]quinoline-4-carboxamide
2-[2-(methoxymethyl)pyrimidin-5-yl]-3,6-dimethyl-4-(pyrrolidine-1-carbonyl)quinoline
[1-(1-cyclopentylpiperidine-4-carbonyl)-3-ethylpiperidin-3-yl]methanol
3-{2-[(4-methoxyphenyl)methyl]morpholine-4-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
(2S)-4-carbamoyl-2-[(3,5,7-trimethyl-1H-indol-2-yl)formamido]butanoic acid
N-(dimethyl-1,2-oxazol-4-yl)-3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)benzamide
1-(cyclohexylmethyl)-3-hydroxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
N'-(2-ethoxyphenyl)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}propanediamide
ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl](quinolin-4-ylmethyl)amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-[5-(thiophen-2-yl)furan-2-yl]propanamide
5-acetyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}thiophene-3-carboxamide
{[2-methyl-1-(2-methylpropyl)-1H-indol-3-yl]methyl}[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]amine
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
1-[(5-{1-[2-(2-hydroxyethoxy)ethyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-ol
6-(1,4-oxazepan-4-ylmethyl)-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2-dihydropyridine-3-carboxamide
1-(cyclopropylmethyl)-5-(2-fluorobenzoyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]butanamide
N-[2-(pyridin-3-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-2,3-dihydro-1-benzofuran-2-carboxamide
2-{1-[1-(2-methoxybenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
2-[2-(4-chlorophenyl)morpholine-4-carbonyl]-3-methyl-1H-indole
1-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(1,3-dimethyl-1H-pyrazol-4-yl)urea
(2R,3S,6R)-5-(cyclopropylmethyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(furan-2-ylmethyl)-1-methyl-3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}urea
5-[4-(1H-pyrazol-1-yl)phenyl]pyridin-2-amine
1-[4-(3-propoxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
2-{[(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}benzoic acid
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
3-[1-(1,3-thiazol-5-ylmethyl)piperidin-3-yl]benzoic acid
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethan-1-one
(3aR,6aS)-1-oxo-5-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-propyl-1H-imidazol-1-yl)-2-(trifluoromethyl)pyridine
4-[3-(pyridin-2-yl)azetidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-amine
6-methyl-8-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
(1R,5S,8S)-8-methoxy-3-(4-methyl-1H-imidazole-2-carbonyl)-3-azabicyclo[3.2.1]octane
8-(2H-1,3-benzodioxole-5-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2,3-difluorophenyl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
pyridin-2-yl({1-[4-(pyridin-3-yl)pyrimidin-2-yl]piperidin-4-yl})methanol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2H-indazol-2-yl)acetamide
{1-[3-(2,4-dimethoxypyrimidin-5-yl)phenyl]ethyl}dimethylamine
1-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
2-{[(4-methoxy-2,3,6-trimethylphenyl)methyl](methyl)amino}-N-methylacetamide