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N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
2-methyl-N-[2-methyl-1-(4-methylpiperazin-1-yl)propan-2-yl]-5-propylpyrimidin-4-amine
3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)pyrrolidine
2-cyclohexyl-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-1,2-dihydroquinoxalin-2-one
2-(2-methoxyethyl)-9-(5-phenyl-1,2,4-oxadiazol-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-4-[(dimethylcarbamoyl)methyl]-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(4-fluorophenyl)-N-[(1s,4s)-4-aminocyclohexyl]imidazo[1,2-a]pyridine-6-carboxamide
6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine-2,4-diamine
(1R,5R)-N,N-dimethyl-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperidine
1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,2,3,4-tetrahydroquinolin-2-one
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
1-(4-methoxyphenyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]cyclopropane-1-carboxamide
1-{4-methyl-2-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]pyrimidin-5-yl}ethan-1-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1H-indole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-(cyclobutylmethyl)-2-(5-ethyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-4-{4-[3-(morpholin-4-yl)-3-oxopropyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-(2-phenyl-1,3-thiazol-4-yl)-N-(pyridin-4-ylmethyl)acetamide
2-(4-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(2-fluorophenyl)methyl]piperazin-2-yl)ethan-1-ol
5-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}quinoline
2-methyl-4-{4-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]phenyl}butan-2-ol
N-[3-(2-ethoxyethoxy)phenyl]-8-methyl-2,8-diazaspiro[4.5]decane-2-carboxamide
(3S,4S)-1-(2-cyanobenzenesulfonyl)-4-propylpyrrolidine-3-carboxylic acid
{3-[(dimethylamino)methyl]-1-(1H-indol-7-ylmethyl)piperidin-3-yl}methanol
1-[2-({[3-(1H-indazol-1-yl)propyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-cyclopropyl-N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)pyrimidine-5-carboxamide
1-phenyl-2-[2-(3-phenylpropyl)morpholin-4-yl]ethane-1,2-dione
3-{1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(2-phenylethyl)piperidine-4-carboxamide
3-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-1-(3-methyl-1-propyl-1H-pyrazol-5-yl)urea
2-(dimethylamino)-1-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]-2-(3-methylphenyl)ethan-1-one
N-[4-(1H-pyrazol-5-yl)phenyl]-1H-indazole-3-carboxamide
ethyl 1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
2,6-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-N-(prop-2-en-1-yl)pyrimidine-4-carboxamide
3-(naphthalen-1-yl)-5-(thiolan-3-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
6-(cyclopropylmethoxy)-4-[2-(1H-imidazol-2-yl)benzoyl]-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
3-[(4-fluorophenyl)formamido]-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]propanamide
3-(benzenesulfonyl)-1-[4-(pyridin-4-yl)piperidin-1-yl]propan-1-one
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(3-fluoropyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-3-(methylsulfanyl)propan-1-one
ethyl 2-{1-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]piperidin-2-yl}acetate
1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-[2-(3-fluorophenyl)ethyl]-N-(1H-imidazol-2-ylmethyl)-6-oxopiperidine-3-carboxamide
2-ethyl-8-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-2-({[4-(3-fluorophenyl)oxan-4-yl]methyl}amino)propanamide
1-(4-{[(1,5-dimethyl-1H-indazol-3-yl)methyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-chloro-4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
ethyl 1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)piperidine-4-carboxylate