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1-benzyl-3-methyl-8-{[3-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
3-methoxy-2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propanoic acid
1-{4-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
N-[2-({[7-chloro-2-oxo-1-(2-phenoxyethyl)-1,2-dihydroquinolin-3-yl]methyl}amino)ethyl]acetamide
2-amino-N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-6-(2-methylpropyl)pyrimidine-4-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-4-(1H-pyrazol-4-yl)butanamide
dimethyl[3-(2-{1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)propyl]amine
7-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxa-7-azaspiro[4.5]decan-8-one
5-(naphthalen-2-yl)-3-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]-1,2,4-triazine
N-{1-oxaspiro[4.5]decan-3-yl}-3-(4H-1,2,4-triazol-4-yl)benzamide
1-(2-methoxy-5-{[4-(propan-2-yl)piperazin-1-yl]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
5-[(1-propyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridazine-4-carboxamide
2-[3-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-oxoacetamide
3-[(2-chlorophenyl)methyl]-5-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazole
N-benzyl-1-(cyclohexylmethyl)-N-(2-hydroxyethyl)-6-oxopiperidine-3-carboxamide
1-(cyclohexylmethyl)-4-oxo-N3-(propan-2-yl)-N5-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
6-[2-(2-{4-[(dimethylamino)methyl]thiophen-2-yl}-1H-imidazol-1-yl)ethyl]pyrimidin-4-ol
2-{4-[(2,5-dimethylphenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
1-[(2,5-dimethylthiophen-3-yl)sulfonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
N-phenyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]pyrimidin-2-amine
methyl 3-acetamido-5-{[(3-methoxyphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-[(2-fluorophenyl)formamido]-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(3S,4S)-4-(naphthalen-2-yl)-1-(pyrimidine-4-carbonyl)piperidin-3-ol
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidine-2-carboxamide
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
6-(2,5-dimethylfuran-3-yl)-2-(3-methoxypiperidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-[(2-fluorophenyl)methyl]-1-(2-hydroxyethyl)-3-[2-(piperidin-1-ylmethyl)phenyl]urea
2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]benzonitrile
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
1-[4-(azepan-1-yl)butyl]-5-oxopyrrolidine-3-carboxylic acid
3-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
4-[2-fluoro-6-(propan-2-yloxy)phenyl]-6-(morpholin-4-yl)pyrimidin-2-amine
2-(3-methyl-1H-pyrazol-1-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
[(3-ethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
3-(4-{7-methylimidazo[1,2-a]pyridin-2-yl}phenyl)-1-(piperidin-4-ylmethyl)urea
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
(3R,4R)-1-(1H-imidazol-2-ylmethyl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
5-(5-fluoro-2-methoxyphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-[(dipropylamino)methyl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-3-sulfamoylthiophene-2-carboxamide
N-(1-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
(2R)-2-cyclohexyl-2-hydroxy-1-{4-[(prop-2-en-1-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
3-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-N-cycloheptylpropanamide
5-methyl-3-(6-methylpyridin-3-yl)-1H-indole