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N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
3,7-dimethyl-11-[4-(1H-pyrazol-5-yl)benzoyl]-3,7,11-triazaspiro[5.6]dodecane
1-cyclopentyl-4-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-one
9-(cyclopropylmethyl)-1-methyl-4-(trimethylpyrimidin-4-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[2-(pyrazin-2-yl)ethyl]acetamide
N-{2-methoxy-4-[2-(prop-2-en-1-ylsulfanyl)propanamido]phenyl}butanamide
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-methylpropanamide
2-{4-[3-(6-hydroxypyrimidin-4-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
2-(butylsulfanyl)-5-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}pyrimidine
methyl 8-(1H-indol-2-ylmethyl)-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl (2S)-1-[5-(2-chloro-4-fluorophenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidine-2-carboxylate
8-[(4-carboxyphenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
(5S,9aS,9bS)-2-[(2-methylphenyl)methyl]-5-(5-methylthiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-cyclohexyl-5-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)pyrimidine
3-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2-methylpyridine
1-[(3S,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
1-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-3-carboxamide
4-(hydroxymethyl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-ol
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-propyl-1,3-oxazole-4-carboxamide
(2S,4R)-4-amino-1-(2-ethoxypyridine-3-carbonyl)-N-methylpyrrolidine-2-carboxamide
3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]-1-[(5-methylthiophen-2-yl)methyl]piperidine
6-{3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]morpholine-4-carbonyl}-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-(1H-1,3-benzodiazol-2-yl)-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}acetamide
2-[(3aS,6aS)-1-[(2-ethylphenyl)methyl]-octahydropyrrolo[3,4-b]pyrrol-5-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
3-{2-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{[1-(dimethylamino)cyclohexyl]methyl}-1,3-oxazole-4-carboxamide
2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-N-methylacetamide
1-[(diethylcarbamoyl)methyl]-N-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-{2-[1-(4-chloro-2-methoxybenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
N-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-N-(3-methylphenyl)methanesulfonamide
(1S,4S)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl)[(5-methylfuran-2-yl)methyl]amine
2-(2,6-dimethoxy-4-methylphenyl)-2-(thiomorpholin-4-yl)acetic acid
7-(2-aminoethyl)-N-(2-methoxyethyl)-N-methyl-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[1-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)piperidin-3-yl]benzoic acid
[1-(1H-indole-5-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-{2-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidin-2-amine
N-[(1R,2S)-2-phenylcyclopropyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
4-(1-benzofuran-2-ylmethyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
(1H-imidazol-2-ylmethyl)[(8-methoxyquinolin-5-yl)methyl]methylamine
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
1-ethyl-3-(3-fluorophenoxymethyl)-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2H-1,3-benzodioxole-5-carboxamide
3-(3-fluorophenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-pyrazole-4-carboxamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide