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1-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
2-[4-(benzyloxy)-2-methylphenyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-[5-({2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
N-[2-(3-methoxyphenyl)ethyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(6-chloropyridazin-3-yl)-N-(1-phenoxypropan-2-yl)piperidin-4-amine
5-(3-acetylphenoxymethyl)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
4-[4-(8-methoxy-2-methylquinolin-5-yl)phenyl]piperidin-4-ol
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
2-(morpholine-4-sulfonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-methyl-N-[3-(4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-2-methyl-1,3-thiazole-4-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-ethyl-3-methylpiperidine-3-carboxamide
2-(3-methoxypropyl)-8-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
2-[methyl({[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]-1-phenylethan-1-ol
4-[1-benzyl-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
(3aR,6aR)-2-(cyclobutylmethyl)-5-(6-ethyl-5-fluoropyrimidin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-3,4-dihydro-2H-1-benzopyran-2-carboxamide
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
(2S,4S)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-[2-(thiophen-3-yl)acetamido]pyrrolidine-2-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(1-methylpiperidin-3-yl)methyl]acetamide
5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
2-methyl-2-(2-{[(2-methylphenyl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
5-(3-acetylphenoxymethyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-methyl-6-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
(2R,6S)-2,6-dimethyl-4-{1-[3-(trifluoromethyl)benzoyl]piperidin-4-yl}morpholine
2-chloro-4-{[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenol
6-[4-(benzylsulfanyl)phenyl]pyrimidin-4-amine
N-ethyl-2-(4-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)acetamide
(2S)-2-{[1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-yl]amino}-3-phenylpropanamide
N-(6-hydroxy-6-methylheptan-2-yl)-2,8-dimethylquinoline-4-carboxamide
4-(1-ethylpiperidin-4-yl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(4-methoxyphenyl)-1-[2-(trifluoromethyl)benzoyl]piperidin-3-amine
3-(1H-pyrazol-3-yl)-N-{2-[2-(pyridin-2-yl)ethyl]phenyl}piperidine-1-carboxamide
1-[(4-fluorophenyl)methyl]-4-[2-(propan-2-yl)-1,3-benzoxazole-5-carbonyl]piperazin-2-one
2-({5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}methyl)-5-methylpyrazine
N-{[(1R,5S,6R)-3-(furan-2-carbonyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}-N-(3-phenylprop-2-yn-1-yl)cyclopropanamine
[(1-ethyl-1H-imidazol-5-yl)methyl][2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]methylamine
{1-[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]piperidin-4-yl}methanol
N-(1-methoxypropan-2-yl)-N-[(2-methylphenyl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[(4-fluorophenyl)methyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
7-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-({6-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyridin-3-yl}methyl)morpholine
1-acetyl-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
N-(3,4-difluorophenyl)-1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
(1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidin-3-yl)methanol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(2-phenoxypyridin-3-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide