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4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-methyl-N-[3-(oxolan-2-yl)propyl]-3-azaspiro[5.5]undecan-9-amine
N-[3-(dimethylamino)-1-phenylpropyl]-8-fluoroquinoline-2-carboxamide
6-methyl-2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carbonitrile
methyl 1-{3-ethyl-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
4-(1-ethyl-1H-imidazol-2-yl)-N,N-dimethylpiperidine-1-sulfonamide
3-phenyl-7-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-(dimethyl-1,2-oxazol-4-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-ethoxyethan-1-one
4-{[4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]methyl}morpholine
2-methyl-N-(1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N,2-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
N-{1-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
4-{[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
N-(3-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl]methoxy}phenyl)propanamide
9-{1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}-6-oxa-9-azaspiro[4.5]decane
1-[(2-fluorophenyl)methyl]-6-oxo-N-[3-(pyridin-3-yloxy)propyl]piperidine-3-carboxamide
4-(4-chlorophenyl)-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)butanamide
1-[(2-chlorophenyl)methyl]-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-(furan-2-ylmethyl)-2-{3-[3-(1-methyl-1H-imidazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
methyl 3-acetamido-1-(oxolan-2-ylmethyl)-5-[(4,4,4-trifluorobutan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-cyclopropyl-2-ethyl-N-({4-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)butanamide
4-hydroxy-2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]quinoline-6-carboxamide
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2-(methylamino)pyridine-4-carboxamide
1-(2-fluorophenyl)-4-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-3-yl)piperazine
2-{[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyrimidine
6-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
3-(2,3-dimethoxy-5-methylphenyl)-6-methylpyridazine
2-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-fluorophenoxy)piperidine
(4aS,8aR)-6-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-(2,2-dimethyloxan-4-yl)-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
methyl 9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate
N-benzyl-3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(3-methylpyridin-2-yl)methyl]propanamide
N,3-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
N-{4-[3-(1-methylpiperidin-3-yl)propanamido]phenyl}pentanamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
1-ethyl-4-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1,2-dihydropyridin-2-one
[(3aS,6aS)-2-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-(cyclopropylmethyl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-chloro-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(furan-2-ylmethyl)-5-{[(2-methoxyphenyl)methyl]amino}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3,5-dimethyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
6-methyl-2-[(4-methyl-1H-imidazol-5-yl)methyl]-5-[5-(oxan-4-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(1H-imidazol-2-ylmethyl)-N-methyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine