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5-{1-[(2,5-dimethoxyphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-tert-butyl-N-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-1,2-oxazol-3-amine
N'-(2-fluoro-5-methylphenyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylbutanediamide
2-amino-6-(4-fluorophenyl)-4-(trimethyl-1H-pyrazol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
methyl 6-(3-phenylprop-2-ynoyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(5-methylfuran-2-yl)methyl]-3-{1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}propanamide
{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
N-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
4-hydroxy-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(3-methylphenyl)pyrimidine-5-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(pyridazine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(1-ethyl-1H-pyrazol-4-yl)-4-(2-ethylmorpholine-4-carbonyl)-6-fluoroquinoline
5-acetyl-N-cyclopropyl-2,4-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrrole-3-carboxamide
5-ethyl-4-[3-(2-methoxyphenoxy)azetidin-1-yl]-2,6-dimethylpyrimidine
N-[2-(2-methoxyphenyl)ethyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(4-fluorophenyl)methyl]-4-methyl-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
ethyl 4-{6,7-dimethoxy-3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}piperazine-1-carboxylate
5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[(3-methylpyridin-4-yl)methyl]amine
(3S)-3-amino-3-{[(2-methoxyphenyl)methyl][(3-methylphenyl)methyl]carbamoyl}propanoic acid
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-7-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide
5-{1-[4-(1H-pyrrol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-[4-phenyl-1-(pyridine-3-sulfonyl)piperidin-4-yl]ethan-1-one
[1-(quinoxalin-2-yl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
2,6-diamino-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
9-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[2-(thiophen-2-yl)ethyl]propanamide
N-(carbamoylmethyl)-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(4-fluoro-3-methylphenyl)-N,N-dimethylpyridine-3-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)propanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-propylpyridine-4-carboxamide
1-[4-(6-aminopyrimidin-4-yl)phenyl]-3-ethylurea
2-(dimethylamino)-2-(4-fluorophenyl)-1-(4-fluoropiperidin-1-yl)ethan-1-one
2-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)amino)-2-[4-(hydroxymethyl)phenyl]acetic acid
N-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-4-(2-methylphenyl)piperazine
N4-ethyl-N2-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}pyrimidine-2,4-diamine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(5S)-5-({[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-2-one
7-(5-ethoxyfuran-2-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(thiophen-3-ylmethyl)piperidin-3-ol
N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,4S)-N-ethyl-4-[2-(2-fluorophenyl)acetamido]-1-(3-hydroxypropanoyl)pyrrolidine-2-carboxamide
6-(2,5-dimethylphenyl)-N-[(1S,2R)-2-hydroxycyclopentyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2,3-dimethyl-6-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}quinoxaline
N-(1,2-oxazol-5-ylmethyl)-3-{[2-(1,3-thiazol-2-yl)ethyl]sulfamoyl}benzamide
2-(1H-pyrazol-3-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
3-methoxy-1-[3-(1H-pyrazol-4-yl)propyl]piperidine