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3-(3-fluorophenyl)-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl][(2,2-dimethyl-1-phenylcyclopropyl)methyl]methylamine
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-ethyl-3-methoxy-N-(2-methylprop-2-en-1-yl)benzamide
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-4-ethyl-1,2,3-thiadiazole-5-carboxamide
4-(4-{1-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]propanamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(2-oxopiperidin-1-yl)propanamide
7-chloro-3-[2-(1-cyclopentylpiperidin-4-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-(1-ethyl-1H-imidazol-2-yl)-1-(3-phenylbenzoyl)piperidine
N-cyclopropyl-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(2-methylpropyl)amine
N-[(3R,4S)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]ethane-1-sulfonamide
N-(furan-2-ylmethyl)-1-(5-methyl-1,2-oxazole-4-carbonyl)piperidine-4-carboxamide
N,N-dimethyl-2-phenyl-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
2-{[(3S,5S)-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-1-[(4-methoxynaphthalen-1-yl)methyl]pyrrolidin-3-yl]sulfanyl}-4,6-dimethylpyrimidine
N-[(8-methoxyquinolin-5-yl)methyl]-N,1-dimethyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[2-(2-methylphenyl)pyrrolidin-1-yl]ethan-1-one
5-(2-chlorophenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]furan-2-carboxamide
5-(oxan-2-yl)-3-(2-phenylethyl)-1H-1,2,4-triazole
N-{[2-(trifluoromethoxy)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]propanamide
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}piperazine
4-(3-hydroxypiperidin-1-yl)-N-(5-methoxy-2-methylphenyl)piperidine-1-carboxamide
1-tert-butyl-4-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(3-methylpyridin-2-yl)piperazine
4-(4-methoxyphenoxy)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
4-{1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}-1-(propan-2-yl)piperidine
5-[4-({[1-(3,5-dimethyl-1H-pyrazol-4-yl)propan-2-yl]amino}methyl)piperidin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-methylpiperidine
3-[(2-fluorophenyl)methyl]-5-(oxan-2-yl)-1,2,4-oxadiazole
4-[2-(pyrrolidin-1-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(2-phenylpropyl)-8-[2-(1H-pyrazol-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-dimethyl-4-[2-(2-phenylphenyl)-1H-imidazol-1-yl]butanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-8-methoxy-3,4-dihydroquinazolin-4-one
N-butyl-1-[2-(3-chlorophenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
4-({2-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperazine-2-carboxylic acid
3-fluoro-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-(piperidin-1-yl)butanamide
1-(piperidin-1-yl)-3-[4-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]propan-2-ol
3,6-dimethyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[(4-ethylphenyl)methyl]-N-(2-methoxyethyl)-1,4-dioxane-2-carboxamide
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-butyl-4-[2-(4-methyl-1,4-diazepan-1-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-propanoylpiperidine-3-carboxamide
N-[2-(4-fluorophenyl)ethyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide