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N-[1-(4-chlorophenyl)cyclopropyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
N-cyclooctyl-5-methyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-15-methyl-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
[1-({1-[(8-fluoroquinolin-2-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N6-cyclopropyl-N4-methyl-N4-[2-(pyridin-4-yl)ethyl]pyrimidine-2,4,6-triamine
N4-ethyl-N2,N4-dimethyl-N2-(pyridin-3-ylmethyl)pyrimidine-2,4-diamine
5-methoxy-3-methyl-2-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}-1H-indole
3-(2,4-difluorophenyl)-1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
methyl(3-methylbut-2-en-1-yl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)cyclohexanecarboxamide
2-[4-(1-methylpiperidin-4-yl)piperidin-1-yl]-4-(piperidine-1-carbonyl)pyridine
3-(4-methyl-1H-pyrazol-1-yl)-N-(propan-2-yl)benzamide
(2S)-N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-acetamido-4-(methylsulfanyl)butanamide
[4-(2-phenylethyl)-1-(thiophene-3-carbonyl)piperidin-4-yl]methanol
2-(3-methylbut-2-en-1-yl)-8-[(3-phenyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-(quinolin-6-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
6-(8-methoxy-2-methylquinolin-5-yl)-1,2,3,4-tetrahydroquinazoline-2,4-dione
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methylphenyl)-1,4-diazepane
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(4-hydroxypiperidin-1-yl)ethan-1-one
4-(1H-indol-4-yl)-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N-ethyl-N-methyl-2-[1-(1-methylpiperidin-4-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-methyl-3-{2-[4-(pyrimidin-2-yloxy)phenyl]-1H-imidazol-1-yl}benzamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]cyclohexanecarboxamide
4-(2-aminopyridin-3-yl)-N-benzylbenzene-1-sulfonamide
1-methyl-4-{[4-methyl-5-(1-methylpiperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
2-(2-{[(1-hydroxycyclohexyl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
3-tert-butyl-1-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
methyl 3-(2-chlorobenzoyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-cyclopropyl-3,5-dimethyl-N-(thiophen-3-ylmethyl)-1H-indole-2-carboxamide
1-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]piperazine
ethyl 4-[({2-[benzyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)amino]piperidine-1-carboxylate
3-chloro-N-(3-cyclopentylpropyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
[5-({ethyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-(propan-2-yloxy)phenyl]methanol
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}pent-4-en-1-one
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridine-3-carbonitrile
5-[4-(furan-2-ylmethyl)piperazine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
1-[(1-{furo[3,2-c]pyridin-4-yl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methylbenzamide
1-[(2R)-2-amino-3-methylbutanoyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
(3S,4R)-4-(3-fluorophenyl)-1-[(4-methanesulfonylphenyl)methyl]pyrrolidine-3-carboxylic acid
5-(1H-indol-1-ylmethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
(3S,4S)-4-(dimethylamino)-1-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
2-amino-6-[4-(morpholin-4-ylmethyl)thiophen-2-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
4-fluoro-N-(2-{[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-5-yl]formamido}ethyl)benzamide
({5-[1-(4-ethoxybenzoyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-[2-(1-hydroxycyclopentyl)ethyl]pyridine-4-carboxamide
(3E)-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylpent-3-enamide