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6-{4-[(3-chloro-2,4-difluorophenyl)methyl]piperazin-1-yl}pyridine-2-carbonitrile
3-(2-methoxyethyl)-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-3-(thiophen-2-ylmethyl)urea
2,5-dimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1,3-thiazole-4-carboxamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-(propan-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-methyl-4-[5-(oxolan-3-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
3-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-2-methylphenol
1-[3-(4-cyclopropanecarbonylphenyl)propyl]-1H-imidazole
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl}){[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amine
3-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
(1S,5R)-3-benzyl-6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-(1,3-benzothiazol-2-yl)-4-(3-chlorobenzenesulfonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-({1-[(2,6-dichlorophenyl)methyl]pyrrolidin-3-yl}methyl)cyclopropanecarboxamide
2-(morpholin-4-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}benzamide
4-[(4-chloro-3-fluorophenyl)methyl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
methyl 4-({2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamido}methyl)benzoate
2-[4-(pyrimidin-2-yl)-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenoxy]-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
(3R,4R)-1-(2-methylfuran-3-carbonyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-cyclohexanecarbonyl-4-[2-(4-fluorophenoxy)ethyl]-1,4-diazepan-5-one
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
4-(thiophen-2-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}butanamide
N-methyl-2-[2-(4-phenyl-1H-imidazol-1-yl)phenoxy]acetamide
N-[(3-methoxyphenyl)methyl]-5-methyl-6-(4-methyl-1,4-diazepane-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-[(4-chlorophenyl)(phenyl)methyl]-1-[1,3-dioxo-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
1-[(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
6-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
(3aS,6aS)-2-[(1,3-dimethyl-1H-pyrazol-5-yl)sulfonyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(butan-2-yl)-2-(2,5-dimethoxyphenyl)-N-(pyridin-4-ylmethyl)acetamide
2-methyl-8-[2-methyl-2-(4-methylphenoxy)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
N-[4-(3-methoxyphenyl)phenyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidine-2-carboxamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]cyclobutanecarboxamide
N-methyl-N-(2-phenyl-1-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl)pyridine-2-carboxamide
1-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,3-diethylurea
ethyl 1-{3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanoyl}piperidine-3-carboxylate
N-[(3S,4R)-1-(butane-1-sulfonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
2-[4-(piperidin-3-yl)benzoyl]-2,3-dihydro-1H-isoindole
2-{4-[1-(2-methoxyphenyl)piperidin-4-yl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
[(1-cyclopentylpiperidin-4-yl)methyl][(2-ethoxyphenyl)methyl](oxolan-2-ylmethyl)amine
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
(3R,4S)-4-cyclopropyl-1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-amine
N-(2H-1,3-benzodioxol-4-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
methyl 3-(2-phenylacetamido)-5-[(1,3-thiazol-5-ylformamido)methyl]benzoate
1-(4-{4-chloro-2-[4-(cyclopropylmethyl)piperazine-1-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
4-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-methyl-1-propyl-1H-pyrazole
ethyl N-{[(2S,4S)-4-fluoro-1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]pyrrolidin-2-yl]methyl}carbamate
1-(5-{[(3S,4S)-3-hydroxy-4-[4-(pyrazin-2-yl)piperazin-1-yl]pyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
[(3-fluoro-2-methoxyphenyl)methyl](methyl)[(1-methylpiperidin-2-yl)methyl]amine
7-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-2-(cyclopropylmethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one