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N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-4H-chromene-3-carboxamide
5-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}pent-4-enamide
2-methyl-6-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]pyrimidin-4-ol
(3S,4S)-1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-N-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3-carboxamide
2-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
4-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-3-yl}benzoic acid
(2-{2-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-{2-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl}pyridin-3-amine
methyl 1-(3-{4-[(tert-butylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
3-(3-aminopyrrolidine-1-carbonyl)-N-(oxan-4-ylmethyl)benzene-1-sulfonamide
5-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-N-cyclopentyl-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-cyclopropyl-N-[3-(dimethylamino)-2,2-dimethylpropyl]-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
4-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine
(2R,3S,6R)-3-(4-methylphenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 1-(2-methoxyethyl)-5-[(5-methylhex-5-en-2-yl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 6-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-[(4-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aR,7aS)-1-benzyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
2,4,5-trimethyl-6-{4-[(methylsulfanyl)methyl]piperidin-1-yl}pyrimidine
1-cyclopentyl-4-oxo-N-(prop-2-en-1-yl)-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-phenyl-1-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethan-1-one
N-methyl-N-[(5-methylfuran-2-yl)methyl]-3-sulfamoylthiophene-2-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
1-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazol-3-yl)ethan-1-one
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-2H-chromene-3-carboxamide
3-propyl-1-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]urea
2-methyl-N-{1-[7-(quinolin-7-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
[4-(2-methyl-4-phenylpyrimidine-5-carbonyl)-1,4-oxazepan-6-yl]methanol
1-[(2,3-difluorophenyl)methyl]-5-{2-[(2-methoxyethyl)amino]ethyl}pyrrolidin-2-one
methyl 2-({5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl}formamido)-2-methylpropanoate
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}cyclobutanecarboxamide
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-3-methylthiophene-2-carboxamide
4-[2-(4-fluorophenyl)acetyl]-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
5-chloro-2-(oxolan-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline
N-{2-[1-(3-chloro-2-methylbenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
9-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(1H-indol-3-yl)-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}propan-1-one
2-{[4-(1,5-dimethyl-1H-indazol-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
(3aR,6aS)-5-(1,1-dioxo-1λ6-thiane-4-carbonyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(1R,3S)-3-[4-(hydroxymethyl)piperidine-1-carbonyl]cyclopentyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-[2-(4-methoxyphenyl)phenyl]-1-(pyridine-4-carbonyl)pyrrolidine-2-carboxamide
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}thiolan-3-amine
N-[(3-methyloxetan-3-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
methyl[1-(1,2-oxazol-3-yl)ethyl]{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-methyl-6-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-3,4-dihydroquinazolin-4-one