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methyl 2-(tert-butylsulfamoyl)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl})amine
2,5-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-(4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}benzamido)benzamide
6-methoxy-1-methyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-indole-2-carboxamide
5-({3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-3-carboxamide
7-(2-methoxyethyl)-2-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-butyl-5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
1-[1-(3-hydroxypropanoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
2-(3-chloro-4-hydroxyphenyl)-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
N-butyl-3-[(cyclobutylamino)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
3-chloro-2-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
{1-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
2-methoxy-N-(1-{1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-methyl-N-[3-(3-methylphenoxy)propyl]-2-(phenylamino)pyrimidine-5-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(6-methylpyridin-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1,3-dimethyl-N-[4-(pyrrolidin-1-yl)butyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(2,3-dihydro-1H-inden-2-yl)-4-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazine
5-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-{2-[(3,3-dimethylcyclohexyl)amino]ethyl}-N-methylmethanesulfonamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(methylamino)pyridine-3-carboxamide
1-[2-({1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]piperidin-2-one
6-methoxy-4-[2-(1H-pyrazol-1-yl)benzoyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
2-({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)propane-1,3-diol
4-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[2-(2-methoxyphenyl)ethyl]-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
1-{1-[(2Z)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-3-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine-3-carboxylic acid
N-[3-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)carbamoyl}methoxy)phenyl]propanamide
2-methoxy-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)piperidin-2-one
(3aS,6aR)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-ethyl-3-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-fluorophenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-pyrazole-4-carboxamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(2-methoxyacetyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}piperidine-4-carboxamide
2-ethyl-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
2-(methoxymethyl)-1-[(5-methylthiophen-2-yl)methyl]piperidine
7-(1,3-benzothiazol-2-yl)-4-benzyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S)-1-acetyl-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
5-hydroxy-N-{5-[2-(4-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}pyrazine-2-carboxamide
5-({spiro[azepane-4,2'-chromene]-1-yl}carbonyl)pyridine-2-carbonitrile
(2S,4S)-4-(5-methyl-1-propyl-1H-pyrazole-4-amido)pyrrolidine-2-carboxylic acid
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(3aS,6aS)-2-[(2-fluoro-4-methoxyphenyl)methyl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-hydroxy-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methylbenzamide