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N-methyl-N-(quinoxalin-2-ylmethyl)quinoxaline-2-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-(1H-pyrazol-1-yl)benzene-1-sulfonamide
(1S,5R)-3-[(4-acetylphenyl)methyl]-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
6-{[(2,2-dimethylcyclopentyl)amino]methyl}-2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)-3,4-dihydropyrimidin-4-one
N-[(2S,4R,6S)-2-(1-ethyl-1H-imidazol-5-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
methyl (2S,4R)-1-methyl-4-[(E)-2-phenylethenesulfonamido]pyrrolidine-2-carboxylate
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-ethyl-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
methyl (2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
2-(3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl)-4H-chromen-4-one
(1S,5R)-N-benzyl-6-[(dimethylcarbamoyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3aR,6aR)-2-[2-(4-fluorophenyl)ethyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(dimethylamino)propan-2-yl]-2-methyl-1-benzofuran-5-carboxamide
4-[2-(2-oxopyrrolidin-1-yl)acetyl]-1-(2-phenylphenyl)piperazin-2-one
N-[4-(furan-2-yl)phenyl]-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidine-3-carboxamide
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(1H-pyrazol-1-ylmethyl)piperidine-1-carboxamide
2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-6-methylpyridine-3-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(thiophen-3-yl)acetamide
1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(4H-1,2,4-triazol-4-yl)piperidine
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
1'-(benzenesulfonyl)-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
2-{[6-(5-fluoro-2-methylphenyl)pyridazin-3-yl]amino}ethan-1-ol
4-benzyl-3-ethyl-1-(2-methoxypyrimidine-5-carbonyl)-1,4-diazepan-5-one
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(3-methoxypropyl)benzamide
1-[4-({[(3,5-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
(1R,9aR)-1-({[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
2-{1-benzyl-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-(3-methylbutyl)-3-{2-oxo-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}piperazin-2-one
4-{[ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})amino]methyl}-2,6-dimethoxyphenol
1-[2-(4-fluorophenyl)morpholin-4-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
(1R,5R)-6-(2-methoxyethyl)-3-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-cyclobutanecarbonyl-3-(2-phenylethyl)piperidine
1-methyl-2-oxo-8-[2-(thiophen-2-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(6-methylquinolin-4-yl)-decahydro-1,6-naphthyridin-2-one
4-(1-benzothiophen-2-ylmethyl)morpholine-2-carboxylic acid
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]ethyl]methylamine
3-{[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzonitrile
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
1-{2-[4-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2,3-dimethyl-7-{[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1H-indole
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-cyclopentyl-3-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)urea
N-benzyl-6-[(2E)-3-phenylprop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
propyl 4-{[4-(pyridin-3-yloxy)phenyl]carbamoyl}piperidine-1-carboxylate
methyl 1-[(3R,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-[(2-hydroxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[3-methyl-4-({methyl[(2E)-3-phenylprop-2-en-1-yl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
2-methyl-4-(3-methyl-5-{2-methylimidazo[1,2-a]pyrimidin-3-yl}-1H-1,2,4-triazol-1-yl)pyridine
(3E)-N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pent-3-enamide
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
N-tert-butyl-3-[3-(3-hydroxy-1,2-oxazol-5-yl)propanamido]-2-methylbenzamide