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2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(piperidine-1-carbonyl)pyrazine
5-(methoxymethyl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}furan-2-carboxamide
methyl 2-(5-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
[7-(4,6-dimethoxypyrimidin-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
2-{4-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-benzyl-N5-ethyl-N3-methyl-4-oxo-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-(6-carbamoylpyrazin-2-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-[(3S,4R)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[(5-methyl-1,2-oxazol-3-yl)methyl]cyclopentane-1,3-dicarboxamide
5-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]pyridin-2-amine
2-{2-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
N-{1-[1-(3-chlorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(2S)-2-amino-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(4-hydroxyphenyl)propan-1-one
N-[(3S,4R)-4-propyl-1-(2,4,5-trimethoxybenzoyl)pyrrolidin-3-yl]acetamide
2-(4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
3-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3-carbonyl}pyridine
6-{[1-(morpholin-4-yl)cycloheptyl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
methyl 6-(3-fluorobenzoyl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
{[4-(3-chlorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
4-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]-1λ6-thiane-1,1-dione
4-{2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
3-(2,5-dioxoimidazolidin-4-yl)-N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]propanamide
ethyl 3-{[1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
2-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-N-methylpyridine-3-carboxamide
5-({3-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
1-(2-hydroxy-3-{4-methoxy-2-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propyl)piperidin-4-ol
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(methanesulfonylmethyl)piperidine
(2R,3R)-3-(dimethylamino)-1'-(1-methyl-1H-pyrrole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(2-chloro-4-fluorophenyl)methyl]-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
4-({5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
ethyl 3-[(4-fluorophenyl)methyl]-1-(2-methoxyacetyl)piperidine-3-carboxylate
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-benzyl-N-butyl-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-methoxyphenyl)ethan-1-one
1-(2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}pyrimidin-4-yl)piperidin-4-ol
(3R,4R)-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-[(3-fluorophenyl)methyl]-4-(6-methyl-1,3-benzothiazol-2-yl)piperazin-2-one
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}azepan-2-one
4-[(3S,5R)-5-[4-(1H-pyrazol-3-yl)piperidine-1-carbonyl]piperidine-3-carbonyl]morpholine
N4-{2-[(3-methylpyridin-2-yl)amino]ethyl}-6-(propan-2-yl)pyrimidine-2,4-diamine
3-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
6-[3-(4-chlorophenyl)piperidine-1-carbonyl]-2-cyclopropyl-1,3-benzoxazole
3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-3-yl}benzoic acid
(1R,5R)-6-benzyl-3-(1-methyl-1H-indole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane