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N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-6-oxopiperazine-2-carboxamide
methyl 1-[(3R,5S)-1-[(2,4-dimethylphenyl)methyl]-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[(1-ethyl-1H-indazol-3-yl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
(1R,2S,4R)-N-butyl-N-(thiophen-3-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
methyl 3-benzamido-5-{[(5-ethylfuran-2-yl)methyl]amino}-1-(furan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-methoxy-2-[4-(2-phenylethyl)piperidine-1-carbonyl]-4H-pyran-4-one
2-acetyl-8-(4-carboxy-1,3-oxazol-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{4-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexane-3-carbonyl]phenyl}phenol
1-(1,4-oxazepan-4-yl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
N-(carbamoylmethyl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
N-{[(3S,4S)-1-(1H-1,3-benzodiazole-5-carbonyl)-3-hydroxypiperidin-4-yl]methyl}furan-2-carboxamide
N-(butan-2-yl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
2-{[methyl({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl})amino]methyl}benzonitrile
4-methyl-2-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
1-(2-oxo-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydroquinolin-2-one
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
[4-(2-phenylethyl)-1-[4-(piperidin-1-yl)benzoyl]piperidin-4-yl]methanol
9-methoxy-N-(3-methylbutyl)-7-oxo-3-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(4-cyano-2-ethylphenyl)-3-{[4-(dimethylamino)oxan-4-yl]methyl}urea
(1R,4S)-1,7,7-trimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
N-(1-hydroxybutan-2-yl)-3-(1H-pyrazol-1-ylmethyl)-N-(pyridin-3-ylmethyl)benzamide
1-{1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]piperidin-4-yl}-2-phenylethan-1-ol
6-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
1-methyl-6-(pyridin-4-yl)-N-(thiolan-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-ethoxy-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{[7-chloro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-1,3-thiazole-5-carboxamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-3-(4-methylphenyl)-1H-pyrazole-5-carboxamide
N-({8-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methylpropanamide
butyl (2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
3-(3-fluorophenyl)-N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-1H-pyrazole-4-carboxamide
N-benzyl-N-ethyl-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenoxyacetamide
2-[3-methyl-5-(3-methyl-1,2-oxazol-5-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
1-(cyclohexylmethyl)-N-(cyclopropylmethyl)piperidin-3-amine
5-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)-2,1,3-benzothiadiazole
N-(oxolan-2-ylmethyl)-7-(1H-pyrazole-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[3-({ethyl[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenyl]-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
3-chloro-2-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}pyridine
N-({7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
methyl({[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl})(quinoxalin-2-ylmethyl)amine
methyl 5-{[(2,5-dimethylphenyl)methyl]amino}-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2R,3R)-1'-(3-chlorothiophene-2-carbonyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
8-(1H-imidazole-2-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-methyl-1-(1-{6-[(pyridin-3-ylmethyl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
2-{5-[5-(1H-imidazol-1-ylmethyl)furan-2-yl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-ethoxypropyl)acetamide
4-{1-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenol