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1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
6-{6-hydroxy-4-[2-(1H-imidazol-1-yl)acetyl]-1,4-diazepan-1-yl}pyridine-2-carbonitrile
3-[2-(benzyloxy)ethyl]-4-methoxybenzamide
2-(dimethylamino)-N-methyl-N-(pyrazin-2-ylmethyl)benzamide
1-{1-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
(3-{2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
ethyl 1-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1H-imidazole-2-carboxylate
2-(cyclopropylmethyl)-9-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-fluorophenyl)-4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]morpholine
2-{4-[2-(1H-imidazol-1-yl)acetyl]morpholin-3-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
2-[4-(5-chloro-2-methoxypyridin-4-yl)phenyl]-N-methylacetamide
N'-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N'-[2-(4-fluorophenyl)ethyl]-N,N-dimethylbutanediamide
6-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5R)-6-(2-{[(4-chlorophenyl)methyl]carbamoyl}ethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
8-[3-(pyridin-4-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-N-(oxan-2-ylmethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-4-methylphenol
(isoquinolin-5-ylmethyl)(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
3-chloro-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]thiophene-2-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[2-(thiomorpholin-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}morpholine-4-sulfonamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,3-oxazole-5-carbonyl)piperidin-3-ol
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-methylfuran-3-carboxamide
(2E)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
N-{[4-(prop-2-en-1-yl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}-2-(trifluoromethyl)benzamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyrazine
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(7-methyl-2-oxo-2H-chromen-4-yl)acetamide
5-[methyl(2-phenylethyl)amino]-2-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]propanamide
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-[3-(pyridin-3-yl)propyl]pyrrolidin-3-yl]sulfamoyl})amine
1-{[2-(3-chlorophenyl)-6,7-dimethoxyquinolin-3-yl]methyl}piperidine-3-carbonitrile
(1S,9S)-11-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-[3-(4-{[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
(4aS,8aR)-6-[(3-chlorophenyl)methyl]-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
N-(1,4-dioxan-2-ylmethyl)-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
1-(3,4-dimethylphenyl)-3-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-[methyl(propan-2-yl)amino]propan-1-one
1-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(pyrimidin-2-yl)ethan-1-one
6-ethyl-2-methyl-N-(oxan-4-yl)quinoline-4-carboxamide
2-methyl-3-[4-(2-methylphenoxy)piperidine-1-carbonyl]-2,8-diazaspiro[4.5]decane
7-(2,2-dimethylpropyl)-2-[(5-methylfuran-2-yl)methyl]-2,7-diazaspiro[4.5]decane
1-(azocan-1-yl)-3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-one
2-methyl-1-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)azetidin-3-yl]piperidine
N-methyl-4-(piperidin-3-ylmethyl)-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine