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1,8-dimethyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(pyridin-2-ylsulfanyl)acetamide
2-benzyl-8-(6-cyclopropylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(4-ethylmorpholin-2-yl)ethyl]-3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carboxamide
N-(propan-2-yl)-1-(2-{1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
methyl 3-(2,1,3-benzothiadiazol-5-ylmethyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-cyclopropyl-N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
(4aR,8aR)-2-(3,6-dimethylpyrazin-2-yl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
3-{4-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}propan-1-ol
N-(2-chlorophenyl)-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-chloro-2-[2-(1H-imidazol-2-yl)-1H-pyrrol-1-yl]pyridine
1-[(1S)-1-[1-(3-chloro-4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl]-1H-1,2,3,4-tetrazole
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-4-yl)propan-1-one
3-{[(2-hydroxyphenyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-methoxy-N-({1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-[(4-fluorophenyl)methyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
4-(2-ethyl-1-benzofuran-3-yl)-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
(1R,5R)-6-(2,3-dihydro-1H-indene-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-(1-benzofuran-2-yl)-3-methylpyridin-2-amine
N-(3-hydroxypropyl)-2-methyl-N-[(5-methylthiophen-2-yl)methyl]butanamide
{1-[(E)-2-phenylethenesulfonyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-2-[(3-methoxyphenyl)methyl]morpholine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
2-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-indole
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-4-(piperidin-1-ylmethyl)benzamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
2-(3-cyanophenyl)-N-propylbenzamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl]propanoic acid
2-(methylamino)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)benzamide
N-[2-(4-fluorophenyl)-1-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl]-2-methoxy-N-methylacetamide
1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
3-(pyridin-3-yl)-N-({7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)propanamide
2-(cyclopropylmethyl)-7-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-[({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)methyl]-1λ6-thiolane-1,1-dione
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-methyl-6-(4-methylphenyl)-N-[3-(morpholin-4-yl)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-({4-[(3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
4-(1H-imidazol-1-ylmethyl)-1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-ol
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(3-methoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
N-[2-(methylsulfamoyl)ethyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
N-(butan-2-yl)-2-chloro-4,5-difluoro-N-(pyridin-4-ylmethyl)benzamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-3-carboxamide
3-{1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}pyridine