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1-({4-methyl-5-[1-(pyrazin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
4-hydroxy-N-(3-hydroxypropyl)-2-phenylpyrimidine-5-carboxamide
N-(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
3-(2-methylphenyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-ol
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-propyl-1,2,4-oxadiazole
4-(4-{[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]amino}piperidin-1-yl)-N-(pyridin-3-ylmethyl)benzamide
4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole
methyl 2-chloro-4-{[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]amino}benzoate
2-ethyl-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-(propan-2-yl)piperazine
N4-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidine-2,4-diamine
2-{2-[1-(3-cyano-4,6-dimethylpyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
8-[2-(pyrrolidin-3-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethan-1-one
2-acetamido-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
N-(2,3-dihydroxypropyl)-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-(3,3-diphenylpropyl)-6-[(4-acetamidophenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
methyl 5-{[(4-ethoxyphenyl)methyl]amino}-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4S)-4-amino-1-(2-cyanobenzoyl)-N-methylpyrrolidine-2-carboxamide
2-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-5-yl]-N-methylpyridine-3-carboxamide
1-(carbamoylmethyl)-N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidine-4-carboxamide
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
2-(furan-2-yl)-4-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][4-(1H-pyrazol-1-yl)butan-2-yl]amine
1-(2,4-dimethylphenoxy)-3-[(pentan-3-yl)amino]propan-2-ol
2-{1-[(2,2-difluoro-2H-1,3-benzodioxol-4-yl)methyl]azetidin-3-yl}pyridine
1-(2,2-dimethylpropyl)-4-({[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amino)pyrrolidin-2-one
N-[(3R,4S)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-propylpyrrolidin-3-yl]-3-methoxypropanamide
4-[2-(1-methylpyrrolidin-2-yl)ethyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}cyclohexan-1-ol
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
N-[2-(3-hydroxy-4-methoxyphenyl)ethyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
N-methyl-5-{[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]methyl}furan-2-carboxamide
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl})[(3-phenyl-1H-pyrazol-5-yl)methyl]amine
5-(4-methanesulfonylphenyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-methyl-3-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-(4-{4-[(oxolan-2-ylmethyl)amino]piperidin-1-yl}phenyl)-5-phenylpentanamide
N-methyl-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
5-[({[3-(2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
2-(dimethylamino)-N,4-dimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrimidine-5-carboxamide
3-(1-methylpiperidin-2-yl)-N-[3-(1H-pyrazol-1-yl)propyl]propanamide
3-[(2R)-2,3-dihydroxypropyl]-2-oxo-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
[(3R,4S)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-(isoquinolin-5-ylmethyl)-N-methyl-4-(4H-1,2,4-triazol-4-yl)benzamide
2-{[1-(4-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]methyl}morpholine
1-(2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-oxoethyl)piperidin-2-one
(2S,4S)-4-amino-1-{7-amino-2-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide