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5-[(dimethylamino)methyl]-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-2-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(6-methylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
3-(3-chloro-1H-1,2,4-triazol-5-yl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
N-(5-fluoro-2-methylphenyl)-2-{[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}acetamide
N-cyclopropyl-1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-{[6-(5-aminopyridin-3-yl)pyridazin-3-yl](methyl)amino}ethan-1-ol
methyl 4-[3-(2-{[(2,4-dimethoxyphenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]-4-oxobutanoate
(3S,9aR)-8-[(3-methylphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-3-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
1-cycloheptyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
1-methyl-N-[2-(5-methylthiophen-2-yl)ethyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(2-methylpropyl)-5-oxo-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidine-3-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-(1H-pyrazol-3-yl)benzamide
7-[(3E)-hex-3-enoyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl]acetate
2-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
7-(1,3-benzothiazol-2-yl)-4-[(3,4-difluorophenyl)methyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(piperidin-1-yl)ethyl]-3-{[(2S)-pyrrolidin-2-ylmethyl]sulfamoyl}benzamide
1-(furan-3-carbonyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepane
2,5-dimethoxy-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
1-benzyl-4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
6-(2-chlorophenyl)-7-methyl-N-(2-methylbutyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{1-benzyl-4-[(4-ethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2-(2-oxopiperidin-1-yl)acetamide
N-{1-[1-(adamantan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-[2-(4-methoxyphenyl)ethyl]-4-[(propan-2-yl)amino]pyrrolidin-2-one
1-({1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}methyl)pyrrolidin-2-one
8-[(2,4-dimethylphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-phenyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopentyl-4-(2,4-dioxoimidazolidin-1-yl)-N-(3-phenylprop-2-yn-1-yl)benzamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl})amine
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-[(4-methyl-1H-imidazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(1H-imidazol-1-yl)ethyl]-4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-[1-(pyrazin-2-yl)propan-2-yl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl (2S)-1-[2-(4-{4-[(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}phenyl)acetyl]pyrrolidine-2-carboxylate
methyl 4-{[methyl({[2-(pyrrolidin-1-ylmethyl)phenyl]methyl})carbamoyl]amino}benzoate
3-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}-1,2-dihydroquinoxalin-2-one
(4aR,8aS)-1-(2-cyclohexylethyl)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]benzamide
8-{[3-(2-ethyl-1H-imidazol-1-yl)propyl]amino}-2,6-dimethyloctan-2-ol
3-chloro-4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
4-[(4-fluoro-3-methoxyphenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclopropyl-N-{[1-(3,5-dimethylphenyl)cyclopentyl]methyl}-5-oxopyrrolidine-3-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(3-fluoro-4-methylphenyl)methyl]-1,2-oxazole-3-carboxamide
[2-(dimethyl-1,3-thiazol-2-yl)ethyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine