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{3-benzyl-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidin-3-yl}methanol
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)ethyl]amine
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-(2-methyl-1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
N-[(3-fluoro-4-methylphenyl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(1S,5R)-6-benzyl-3-[(3-chloro-1H-indol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-6-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-propyl-decahydro-1,6-naphthyridin-2-one
2-methyl-7-{[5-(1,3-oxazol-5-yl)thiophen-2-yl]sulfonyl}-2,7-diazaspiro[4.5]decane
N-[(3-chlorophenyl)methyl]-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propanamide
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-4-(pyrrolidin-3-yl)benzamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-ethyl-9-{[4-(propan-2-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
2-(2-methoxyethyl)-8-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
2-[(3-benzoylpiperidin-1-yl)methyl]-N-(thiophen-2-ylmethyl)quinazolin-4-amine
2-{4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperazin-1-yl}ethan-1-ol
5-ethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
6-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-2,3-dihydropyridazin-3-one
(3S,4S)-4-methyl-1-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperidine-3,4-diol
8-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
N-cyclopentyl-5-(2,2-diphenylethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(4-{4-[(2-hydroxyethyl)amino]quinazolin-6-yl}phenyl)imidazolidine-2,4-dione
1-(5-propyl-1,2-oxazole-4-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
4-cyclopentyl-3-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}piperazin-2-one
N-methyl-5-{[methyl(2-phenylethyl)amino]methyl}-N-(3-methylbutan-2-yl)-1,2-oxazole-3-carboxamide
{3-[(4-fluorophenyl)methyl]-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl}methanol
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N-methyl-4-oxobutanamide
1-methyl-N-[2-(4-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-4-(pyridin-4-yl)piperidine-1-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[1-(thiophen-3-yl)propan-2-yl]amine
3-(pyridin-2-yl)-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
(1S,5R)-3-(1-benzofuran-5-ylmethyl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(1-{1-[2-(1H-indol-3-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}propyl)acetamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[2-(morpholin-4-yl)propyl]amine
1-[(4-methylphenyl)methyl]-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperazin-2-one
4-[(3-methylpyridin-2-yl)methyl]-N-[4-(methylsulfanyl)phenyl]piperazine-1-carboxamide
5-[7-fluoro-2-({[1-(piperidin-1-yl)cyclohexyl]formamido}methyl)-2,3-dihydro-1-benzofuran-5-yl]pyridine-3-carboxamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(methylsulfanyl)propan-1-one
N-butyl-4-{[(3-fluorophenyl)methyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
15-methyl-13-oxo-N,N-bis(prop-2-en-1-yl)-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-methyl-N-{2-[4-(2-methylpropyl)morpholin-2-yl]ethyl}-1H-pyrazole-5-carboxamide
(3S,4R)-1-cyclopentyl-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
1-{6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]pyrimidin-4-yl}piperidin-4-ol
4-(1H-1,3-benzodiazol-2-yl)-2-chlorophenol
methyl (2S,4S)-1-methyl-4-(6-methyl-2-oxo-1,2-dihydroquinoline-4-amido)pyrrolidine-2-carboxylate
5-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-(2-methoxyethyl)-1,2,4-oxadiazole
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one