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1-(4-fluorophenyl)-4-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butane-1,4-dione
dimethyl({4-methyl-5-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-3-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}urea
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}-2-methanesulfonylacetamide
2-oxo-N-[2-(pyridin-3-yloxy)phenyl]-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
1-ethyl-4-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl]-1H-pyrrole-2-carbonitrile
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
1,3-dimethyl-6-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N'-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N'-methyl-N-(propan-2-yl)ethanediamide
2,3,6-trimethyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
2-(2-{1-[(2,4-dimethylphenyl)methyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
3-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
1-[4-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenyl]imidazolidin-2-one
N-[2-(1-{4-[(4-methylpiperazin-1-yl)methyl]benzoyl}piperidin-2-yl)ethyl]acetamide
1-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazine-1-carbonyl}cyclopropane-1-carboxamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1,2-oxazole-3-carboxamide
9-methoxy-7-(3-methoxyphenyl)-4-[(8-methoxyquinolin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{[2-(3-fluorophenyl)piperidin-1-yl]methyl}pyridin-2-amine
2-(2-{[3-(4-chlorophenyl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
2-methyl-6-{[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
2-(dimethylamino)-2-(3-methylphenyl)-1-(pyrrolidin-1-yl)ethan-1-one
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(1,3-thiazol-2-ylmethyl)pyrimidin-2-amine
7-cyclobutaneamido-N,1-dimethyl-N-[2-(oxan-2-yl)ethyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-{2-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
dimethyl({2-[1-(3-methyl-1,2-oxazole-5-carbonyl)piperidin-2-yl]ethyl})amine
(3S,4S)-1-[3-(2-oxoazepan-1-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
4-chloro-2-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenol
1-methyl-4-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]-1H-1,3-benzodiazole
5-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)furan-2-carboxamide
8-(1,5-dimethyl-1H-indazole-3-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-3-ol
4-{1-[3-(pyridin-2-yl)propyl]-1H-imidazol-2-yl}pyridine
N-(2-chlorophenyl)-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
N-[(1R,2S)-2-phenylcyclopropyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}[(4-fluorophenyl)methyl](prop-2-en-1-yl)amine
(1S,5R)-3-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(dimethylamino)methyl]-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
1-(5-{2-azaspiro[4.4]nonan-2-ylmethyl}-2-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
3-{methyl[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-1-phenylpropan-1-ol
N-[(6-chloro-2H-chromen-3-yl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-[3-(2-phenylethyl)-1,2-oxazole-5-carbonyl]morpholine
1-[3-(2,4-dichlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]piperidine
methyl (2R)-2-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)propanoate
1-(2-methylpropyl)-5-oxo-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-3-carboxamide
methyl[(2-phenyl-1,3-thiazol-5-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine