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1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-cyclopropyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)pyridine-3-carboxamide
2,3-dimethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}quinoxaline-6-carboxamide
N-benzyl-N-methyl-3-{1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-4-yl}propanamide
N-benzyl-1-methyl-N-[(6-methylpyridin-2-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
4-{4-[(2-aminoethoxy)methyl]phenyl}-N,N-dimethylbenzamide
(2R,3S,6R)-3-(4-fluorophenyl)-5-[(2-propylpyrimidin-5-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[2-(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
(2E)-2-methyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)but-2-enamide
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2,2-difluorobutan-1-one
3-({4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]piperazin-1-yl}methyl)piperidin-3-ol
3-(5-methylfuran-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
1-[2-methyl-5-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)phenyl]imidazolidin-2-one
1-[(4-fluorophenyl)methyl]-4-(4-methyl-1H-pyrrole-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
4-(2-methoxyphenoxy)-1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
2-[(3,4-dimethoxyphenyl)methyl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
5-[4-oxo-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridine-2-carbonitrile
1-(azepan-1-yl)-3-{3-[2-(methylsulfanyl)ethyl]-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl}propan-1-one
3-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-(furan-2-ylmethyl)piperidine
N-(2,1,3-benzoxadiazol-4-ylmethyl)-N-methylthian-4-amine
1-ethyl-4-({4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
2-[methyl(pyrazin-2-ylmethyl)amino]-2-[4-(propan-2-yloxy)phenyl]acetic acid
(2-{4-[1-(2,4-dimethylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)urea
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]oxane-4-carboxamide
4-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1λ6-thiomorpholine-1,1-dione
3-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-3-phenylpropan-1-one
1-(4-{[(7-fluoroquinazolin-4-yl)amino]methyl}phenyl)pyrrolidin-2-one
2-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-(1,2-diphenylethyl)-1-(2-methoxyacetyl)piperidine-4-carboxamide
(4aS,8aR)-6-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
7-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,3-diazepane-2,4-dione
2-(ethoxymethyl)-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2S)-2-amino-1-[4-(4-chlorophenoxy)piperidin-1-yl]-3-(1H-imidazol-4-yl)propan-1-one
1-[1-(pentan-3-yl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
7-(cyclopropylmethyl)-N-(furan-2-ylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]benzamide
3-(isoquinolin-5-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-ethyl-3-methyl-1H-pyrazole-4-carboxamide
1-(4-{3-[({[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
3-(hydroxymethyl)-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-3-ol
1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
methyl 6-cyclohexanecarbonyl-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3,5-dimethoxy-2-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzoic acid
7-amino-4-[3-(pyridin-2-ylmethoxy)phenyl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(trifluoromethyl)benzene-1-sulfonamide
5-(methoxymethyl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-{[4-(methylcarbamoyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[5-(methoxymethyl)furan-2-yl]methyl}({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine