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1-(1,4-dioxan-2-ylmethyl)-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[(4-methylphenyl)sulfanyl]piperidine
1-benzyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3S,4R)-1-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-[2-(benzyloxy)ethyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-{3-[2-(morpholin-3-yl)acetamido]propyl}-1,2,5-oxadiazole-3-carboxylic acid
N1-(3-methylpyridin-4-yl)-N2-[4-(propan-2-yl)pyrimidin-2-yl]ethane-1,2-diamine
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-2-propyl-1,3-thiazole
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
5-ethyl-2-[4-({[(3-hydroxyphenyl)methyl](methyl)amino}methyl)phenyl]-6-methyl-3,4-dihydropyrimidin-4-one
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-ol
N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-methyl-N-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]methanesulfonamide
3-{[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzonitrile
4-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide
3-(4-methoxyphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)-1H-pyrazole-5-carboxamide
5-[5-(morpholin-4-ylmethyl)pyridin-2-yl]pyridin-3-amine
3-(azetidine-1-sulfonyl)-N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]benzamide
3-{[1-(1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidin-4-yl]methyl}benzoic acid
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
5-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-2-phenylpyrimidin-4-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-1H-pyrazole-5-carboxamide
(1R,5R)-N,N-dimethyl-6-[(2,3,5,6-tetrafluoro-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(3R,5S)-N-butyl-5-[(4-methylpiperazin-1-yl)methyl]-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
(2S)-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2,3-dihydro-1H-indole-2-carboxamide
2-(3-fluorophenoxymethyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
[3-ethyl-1-(pyrimidin-5-ylmethyl)piperidin-3-yl]methanol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2,8-dimethylquinoline-4-carboxamide
N-phenyl-5-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-{[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
3-{1-[(3,5-dichloropyridin-4-yl)methyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-methyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2E)-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
(1R,3S)-7-[2-(4-chlorophenoxy)ethyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
2-[1-(2,2-dimethylpropyl)-4-[(2-methoxynaphthalen-1-yl)methyl]piperazin-2-yl]ethan-1-ol
1-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}butan-2-ol
1-{[1-tert-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-phenylpyrrolidin-2-one
(4S)-3-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1,3-oxazolidin-2-one
1-[(2,3-difluorophenyl)methyl]-3-[(dimethylamino)methyl]-3-hydroxypiperidin-2-one
1-[(4-cyanophenyl)methyl]-4-phenoxypiperidine-4-carboxylic acid
2-methoxy-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
2-{[1-(5-phenyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]oxy}pyrimidine
(1S,5R)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-[({2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)methyl]-1,2-dihydrophthalazin-1-one
1-(2,2-dimethylpropyl)-4-[2-(4-fluorophenoxy)ethyl]-1,4-diazepan-5-one
2-{5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
5-methyl-1-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-phenylpiperidin-2-one
N-[(2R,3R)-1'-[(2-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]-N-(1,2-oxazol-3-ylmethyl)piperidin-4-amine