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N2,N4-dimethyl-N2-(quinolin-2-ylmethyl)pyrimidine-2,4-diamine
propan-2-yl 4-chloro-3-{[3-oxo-2-(propan-2-yl)piperazine-1-carbonyl]amino}benzoate
methyl 4-{[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]amino}benzoate
1-methyl-3-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
N-methyl-1-(propan-2-yl)-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
N-[(3S,4R)-4-(4-methylphenyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidin-3-yl]acetamide
[(3aS,6aS)-2-(2,3,6-trimethylquinoline-4-carbonyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
6-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(3-fluorophenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)(pyridin-4-ylmethyl)amine
N-(2-methylphenyl)-3-oxo-3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]propanamide
1-{1-[(3-chloro-5-ethoxy-4-hydroxyphenyl)methyl]piperidin-3-yl}pyrrolidin-2-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
4-{4-[(2-hydroxy-4-methoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
5-({3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-2-(trifluoromethyl)pyridine
N-[2-(diethylamino)ethyl]-1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-4-carboxamide
(3S,9aR)-8-(3,5-difluorobenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(4-chlorophenyl)-N-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
2-amino-6-cyclopropyl-4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-[(3-methoxyphenyl)methyl]-N3-[(4-methylphenyl)methyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[1-(oxan-4-yl)piperidine-4-carbonyl]piperidine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-[(3,5-dimethoxyphenyl)methyl]acetamide
5-(1-{2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}piperidin-4-yl)-5-ethylimidazolidine-2,4-dione
1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}-3-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-3-methylurea
1-[(3-methyl-1-benzofuran-2-yl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
ethyl 4-(cyclopropylmethyl)-1-[(4-fluoro-3-methoxyphenyl)methyl]piperidine-4-carboxylate
(2R)-1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]pyrrolidine-2-carboxamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[2-(thiophen-3-yl)acetamido]methyl}benzoate
(1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-3-propylpiperidin-3-yl)methanol
{[1-(piperidin-1-yl)cyclopentyl]methyl}({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
9-(dimethyl-1,3-thiazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(4-hydroxyphenyl)acetic acid
6-methyl-2-(morpholin-4-yl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]pyrimidin-4-amine
1-[3-(3-fluorophenyl)phenyl]-N-(pyridin-4-ylmethyl)piperidin-4-amine
6-chloro-2-(2,3,4-trimethoxyphenyl)-1H-1,3-benzodiazole
4-(4-{[(4,6-dimethylpyrimidin-2-yl)methyl]amino}piperidin-1-yl)-6-ethyl-N,N-dimethylpyrimidin-2-amine
2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazole
2-{1-[(4-fluorophenyl)methyl]-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
(1-{1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanol
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(oxan-2-ylmethyl)amine
1-(2-fluorophenyl)-4-[(3-{[1-(4-methylbenzoyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
methyl (2S,4S)-1-methyl-4-[2-(pyridin-4-yl)ethanesulfonamido]pyrrolidine-2-carboxylate
N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(3-methoxypiperidin-1-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{3-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]phenyl}acetamide