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2-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-2,7-diazaspiro[4.5]decane
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[4-(pyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
5-cyano-N,2-dimethyl-N-{[3-(methylsulfanyl)phenyl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
1-cyclopentyl-4-[4-methoxy-2-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine
N-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-4-[(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]benzamide
1-cyclobutanecarbonyl-3-[2-(2,4-difluorophenyl)ethyl]piperidine
4-(1H-imidazole-5-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-benzyl-3-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}-N-methylpropanamide
N-(2-chlorophenyl)-3-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]propanamide
2-[3-(4-fluorophenyl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-indazol-3-yl)acetamide
2-({5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-4-sulfamoylbenzamide
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-fluorobenzoyl)piperidine
N-(1-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-methoxyacetamide
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-5-methoxy-3,4-dihydroquinazolin-4-one
4-[1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridine
1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
7-fluoro-N-[1-(2-methoxyphenyl)ethyl]-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-(1H-pyrazol-4-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
ethyl 5-(1H-1,3-benzodiazol-2-ylmethyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
1-(2-fluorophenyl)-N-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(2-cyclopropylphenyl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
4'-(cyclobutylmethyl)-3'-oxo-N-propyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-carboxamide
ethyl 4-{[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]carbamoyl}piperazine-1-carboxylate
N-[(1-ethyl-1H-indazol-3-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
methyl 2-{[(3-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](methyl)amino}acetate
[1-(4-fluorophenyl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
2-[ethyl(pyridin-4-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
(1R,5R)-N,N-dimethyl-6-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
N,N-dimethyl-3-[4-(trifluoromethyl)benzoyl]piperidine-1-sulfonamide
2-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
N-[5-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)thiophen-2-yl]acetamide
(3aS,6aS)-2-(2,5-difluorobenzoyl)-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
8-[6-(hydroxymethyl)pyridine-2-carbonyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{[4-methoxy-3-({1-[4-(4-methylphenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}piperazin-1-yl)ethan-1-one
1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-2-{2-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
1-(3,5-dimethylphenyl)-4-(2-methyloxane-2-carbonyl)piperazin-2-one
2-{[4-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}pyridine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
3-methoxy-1-(4-{4-[2-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidin-1-yl)propan-1-one
1-[(2-aminopyridin-3-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
6-(3-chlorophenyl)-N-[(4-fluorophenyl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
{3-[(3-chlorophenyl)methyl]-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl}methanol
2-methyl-6-[7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-4H-3,1-benzoxazin-4-one