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2-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1-oxaspiro[4.4]nonane-4-carboxamide
3-[(dimethylamino)methyl]-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-ol
5-{[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]carbamoyl}-1H-imidazole-4-carboxylic acid
N-(4-{[benzyl(prop-2-yn-1-yl)carbamoyl]methyl}phenyl)butanamide
methyl (2S,4R)-4-(dimethylamino)-1-(2-methylpyridine-3-carbonyl)pyrrolidine-2-carboxylate
6-methyl-1-[(2-methylphenyl)methyl]-3-({[2-(morpholin-4-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-1H-1,2,3-triazole-5-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-(3-ethoxypropyl)-4-(ethylamino)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-{[methyl(6-phenylpyridazin-3-yl)amino]methyl}-3,4-dihydroquinazolin-4-one
N-methyl-2-[(quinolin-8-yloxy)methyl]-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[(3-fluorophenyl)methyl]urea
(4aS,8aS)-2-(4-ethoxybenzenesulfonyl)-decahydro-2,7-naphthyridin-4a-ol
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
7-(3-ethyl-5-hydroxyadamantane-1-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(4-{1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
3-(1H-1,3-benzodiazol-2-ylmethyl)-N-(1H-1,2,3-benzotriazol-5-yl)piperidine-1-carboxamide
4-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-3-carboxamide
(3aR,6aR)-2-(3-cyanopyridin-2-yl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-({1-[6-(piperazin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
3-[(pentan-3-yl)amino]-2,3-dihydro-1λ6-thiophene-1,1-dione
1-methyl-6-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
propan-2-yl 2-chloro-5-[1-(1H-imidazol-1-ylmethyl)cyclopropaneamido]benzoate
2-{3-[4-(morpholin-4-yl)butoxy]phenyl}-1H-1,3-benzodiazole
N-cyclopropyl-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(3-phenylprop-2-yn-1-yl)acetamide
N-ethyl-2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide
2-(1-ethyl-1H-pyrazol-4-yl)-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]quinoline-4-carboxamide
2-{1-benzyl-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-benzyl-9-[2-(2-fluorophenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-[(4-methylphenyl)methyl]acetamide
5-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-3-(2-phenylethyl)-1,2-oxazole
5-cyclopropanecarbonyl-1'-(4-ethylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-(1H-1,2,4-triazol-1-yl)propyl]amine
2-{5-[(2S)-1-benzylpyrrolidin-2-yl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenyl-1,2-dihydrophthalazin-1-one
5-[({[3-chloro-4-(propan-2-yloxy)phenyl]carbamoyl}amino)methyl]-N,N-dimethylfuran-2-carboxamide
N-ethyl-N-[2-(phenylsulfanyl)ethyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3,3,3-trifluoropropan-1-one
N,4-dimethyl-N-[3-(oxolan-2-yl)propyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
6-[3-(furan-2-yl)-3-phenylpropyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-({4-[1-(dimethylamino)ethyl]piperidin-1-yl}methyl)-6-methyl-1,2-dihydroquinolin-2-one
5-methoxy-1-methyl-N-{1-oxaspiro[4.4]nonan-3-yl}-1H-indole-2-carboxamide
5-cyclobutyl-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1,3,4-oxadiazol-2-amine
ethyl 3-[(2-fluorophenyl)methyl]-1-(4,4,4-trifluorobutyl)piperidine-3-carboxylate
3-benzyl-1-methyl-3-[3-(1,4-oxazepan-4-yl)-3-oxopropyl]-2,3-dihydro-1H-indol-2-one
4-methyl-2-(propan-2-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1,3-thiazole-5-carboxamide