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1-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}piperidin-3-ol
5-(2-methylpropyl)-3-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2-oxazole
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-2,3-dimethoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
3-(3-hydroxypropyl)-4-(4-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-benzothiazole-2-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-6-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
5-(5-chloro-2-methoxyphenyl)-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aS,7aR)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2,3-difluoro-4-methoxyphenyl)-5-(2,2-dimethylpropyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-(morpholin-4-ylmethyl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]furan-3-carboxamide
2-[2-(4-fluorophenyl)piperidine-1-carbonyl]-5-methylpyrazine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-2-yl)acetamide
(3S,4S)-4-(4-fluorophenyl)-1-(2-methylpyridine-3-carbonyl)piperidin-3-ol
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2,6-dimethylpyrimidine-4-carboxamide
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-ethoxy-N-[2-(morpholin-4-yl)ethyl]pyrimidin-2-amine
N-(1,1-dioxo-1λ6-thian-4-yl)-N,2-dimethyl-1-benzofuran-5-carboxamide
(1S,2S)-2-{4-[(3-ethyl-4-methyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}cyclohexan-1-ol
3-(5-methyl-1H-pyrazol-1-yl)-1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-pyrrole-2-carboxamide
dimethyl({2-[(oxolan-3-ylmethyl)(thiophen-3-ylmethyl)amino]ethyl})amine
2-{1-[2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carbonyl]piperidin-2-yl}ethan-1-ol
1-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-3-propylurea
N-[2-(2-ethoxyphenoxy)ethyl]-N-methyl-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
3-ethyl-5-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1,2-oxazole-4-carboxamide
1-cyclohexyl-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
3-(2,6-dimethylphenoxy)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)azetidine
2-{[2-(3-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-3-methoxyphenol
2-(4-chlorophenoxy)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(2R,6R)-4-[2-(pyridin-3-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-{3-[3-(2-fluorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
2-{1-cyclopentyl-4-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
1-methyl-4-{[(quinolin-2-yl)amino]methyl}pyrrolidin-2-one
(2S,4R)-4-[(adamantan-2-yl)amino]-1-benzyl-N-methylpyrrolidine-2-carboxamide
2-(methoxymethyl)-1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
3-[(3R,4S)-1-(4,6-dimethylpyrimidin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(4S,4aS,8aR)-4-phenyl-1-(1,3-thiazol-2-ylmethyl)-decahydroquinolin-4-ol
1-(furan-2-ylmethyl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]piperidine-3-carboxamide
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-2-(methylsulfanyl)acetamide
4-[(3,4-difluorophenyl)methyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]piperazin-2-one
1-(4-methoxy-2-methylphenyl)-3-[(5-oxopyrrolidin-2-yl)methyl]-3-(propan-2-yl)urea
1-(1-cycloheptylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-(3,5-dimethoxyphenyl)-2-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)acetamide
5-({2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}methyl)-3-methyl-1,2-oxazole
1-[(3-methoxyphenyl)methyl]-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
1-{4-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]piperidin-1-yl}-2-ethoxyethan-1-one
2-[2-(2-carboxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-1,3-oxazole-4-carboxylic acid
N3-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-N5-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N,N-dimethyl-3-{[2-(pyridin-3-yloxy)propyl]sulfamoyl}benzamide