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1-{1-[(1-ethyl-1H-indol-3-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
N-[(2R,3R)-1'-[3-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-{1-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-4-ol
2-(2-hydroxyethyl)-9-(2-methyl-1-benzofuran-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-ethyl-8-(6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[2-(4-methylphenoxy)ethyl]acetamide
2-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-5,6-dimethylpyridine-3-carbonitrile
2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
3-[1-(2-amino-6-methylpyrimidine-4-carbonyl)piperidin-4-yl]-N-benzyl-N-methylpropanamide
2-(4-{2-[(3-fluorophenyl)methyl]morpholine-4-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
1-[(1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
2-[(3R,4R)-4-(azepan-1-yl)-3-hydroxypiperidine-1-carbonyl]-1,4-dihydroquinolin-4-one
6-fluoro-2-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}amino)methyl]quinolin-4-ol
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]methanol
N-[(3R,4S)-4-cyclopropyl-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]pyrrolidin-3-yl]cyclohexanecarboxamide
1-methyl-3-(4-phenyl-1,2,3-thiadiazol-5-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
3-{1-[(3,5-dimethylphenyl)methyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]methanesulfonamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1H-pyrrole-2-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-[4-(propan-2-yloxy)benzoyl]piperidine
N,N-dimethyl-5-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyridin-2-amine
4-hydroxy-2-(4-methylphenyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrimidine-5-carboxamide
4-(5-chlorothiophen-2-yl)-7-(dimethylamino)-1,2,3,4-tetrahydroquinolin-2-one
4-(2-methylphenoxy)-1-(6-methylpyridine-2-carbonyl)piperidine-4-carboxylic acid
1-cycloheptyl-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidin-2-one
(1S,5R)-3-methyl-6-[(3-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(3-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethoxy}phenyl)propanamide
6-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-2-methyl-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
1'-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{3-[(3-chlorophenyl)methyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methanol
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1-(9H-purin-6-yl)piperidin-4-amine
2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-(thiophen-2-ylmethyl)acetamide
4-(2,4-difluorophenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-chloro-N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3,3-dimethyl-1-({5-[(1-propyl-1H-imidazol-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
7-[3-(2-ethoxyethyl)-1-methyl-1H-1,2,4-triazol-5-yl]-2,3-dimethyl-1H-indole
3-{4-[5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
2-methoxy-N-[(3R,5S)-5-(methylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]pyridine-3-carboxamide
(1S,5R)-6-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
5-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]-2-(4-methyl-1H-pyrazol-1-yl)acetamide
2-{1-benzyl-4-[(3-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(oxolan-3-yl)acetamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-{[3-(2-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]sulfonyl}pyrrolidine
1-[(2R)-2-amino-3-phenylpropanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl (1R,3S,3aR,6aS)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-3-(pyridin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate