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3-methyl-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]furan-2-carboxamide
{4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
1-(cyclohex-3-ene-1-carbonyl)-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
8-[4-(1H-indol-3-yl)butan-2-yl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(propan-2-yl)-1H-1,3-benzodiazole
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(4-{1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}piperazin-1-yl)ethan-1-ol
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(pyridin-2-yl)propan-1-one
4-methoxy-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidin-2-amine
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-1-methylpiperidine-2-carboxamide
1-(3,3-diphenylpiperidin-1-yl)-2-(2-methoxyethoxy)ethan-1-one
(4aR,8aR)-4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-octahydro-2H-1,4-benzoxazine
5-acetyl-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylthiophene-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
3-(furan-2-yl)-1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)propan-1-one
2-methoxy-N-[1-(2-phenylethyl)-7-(4-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
N-[(4-methoxyphenyl)methyl]-N-methyl-2-phenylpyrimidine-5-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-3-amine
1-(carbamoylmethyl)-N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
5-tert-butyl-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,3,4-oxadiazol-2-amine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-methyl-14-[4-(1H-pyrazol-1-ylmethyl)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-acetyl-8-[2-(3-hydroxyphenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
N-[(3S,4R)-4-propyl-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}pyrrolidin-3-yl]acetamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-methoxy-N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane
N-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
3-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-(2-{1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
3,6-dimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1-benzofuran-2-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-(3-fluoro-2-methylphenyl)-2-[3-(2-methoxyphenoxy)azetidin-1-yl]acetamide
1-[4-(adamantan-1-yl)piperazin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-(1H-1,3-benzodiazol-1-yl)-N-{[2-(dimethylamino)pyridin-3-yl]methyl}propanamide
2-[5-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-methyl-1H-1,3-benzodiazole
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N,5-dimethyl-4-phenyl-N-(pyrazin-2-ylmethyl)thiophene-3-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(dimethylamino)-2-methylpropan-1-one
2-amino-8-[1-(oxan-4-yl)piperidine-3-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
(3aS,6aR)-5-(1H-imidazol-2-ylmethyl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-(1-propyl-1H-1,2,4-triazol-5-yl)-2-(pyridin-4-yl)pyrimidine
4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyridine
N-ethyl-3-fluoro-5-methyl-N-[2-(morpholin-4-yl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
4-[6-(1-hydroxyethyl)pyridin-2-yl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-(piperidin-1-yl)propan-2-ol