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6-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(1H-pyrrol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
N-(2-methoxyethyl)-3,5-dimethyl-N-(1-methylpiperidin-4-yl)-1-benzofuran-2-carboxamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[1-(pyridin-4-yl)propyl]benzamide
{3-[(3-chlorophenyl)methyl]-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}methanol
4-{4-[(2-ethoxyphenyl)methyl]piperazin-1-yl}-5-ethyl-2-methylpyrimidine
4-(dimethylsulfamoyl)-N-(2-methylquinolin-8-yl)piperazine-1-carboxamide
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-6-(2-fluorophenyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
9-[2-(3-chloro-4-fluorophenoxy)acetyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(cyclohexylmethyl)-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
[1-(4-methylquinolin-2-yl)-4-(oxan-2-ylmethyl)piperidin-4-yl]methanol
3-(1-butyl-1H-imidazol-2-yl)-1-[2-(1H-pyrazol-1-yl)benzoyl]piperidine
1-{2-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
4-[4-(2-methoxyphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
N-(3-chlorophenyl)-2-[2-(dimethylamino)ethyl]morpholine-4-carboxamide
2-(4-chlorophenyl)-8-[(4-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-(2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}ethyl)phenol
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-{2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
N-[(2R,3R)-2-ethoxy-1'-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-4-(1H-imidazol-2-yl)piperidine
2-(1-butyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
1-phenyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(3-methoxypropanoyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
1-(azepan-1-yl)-3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propan-1-one
1-[(3-methylpyridin-2-yl)methyl]-4-[(5-propylfuran-2-yl)methyl]piperazine
N4-[4-(2-fluorophenoxy)phenyl]-N1,N1-dimethylpiperidine-1,4-dicarboxamide
ethyl 1-(5-acetylthiophene-3-carbonyl)-3-benzylpiperidine-3-carboxylate
N3-butyl-N5-[(2,6-difluorophenyl)methyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-(4-methoxyphenyl)ethyl]-N-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
8-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-[2-(2-hydroxyethoxy)ethyl]-2-methyl-1-benzofuran-7-carboxamide
(3S,7S,8aS)-7-{[(3,4-dimethylphenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-[2-(3-phenylpropyl)morpholin-4-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
(2,1,3-benzoxadiazol-5-ylmethyl)({[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
5-methanesulfonyl-1'-(1-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{2-[4-(6-chloropyridin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}aniline
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]benzamide
3-chloro-N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}benzamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-4-(piperidin-1-yl)butanamide
methyl 1-[2-hydroxy-3-(3-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
N-[(5-chlorothiophen-2-yl)methyl]-1-(9H-purin-6-yl)piperidin-4-amine
4-acetyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
2-(1-methyl-1H-pyrrol-2-yl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-2-oxoacetamide
7-fluoro-2-methyl-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]quinoline-4-carboxamide
(1R,5R)-6-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane