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N-{[5-(1H-imidazol-2-yl)furan-2-yl]methyl}-N-methylmethanesulfonamide
N-(4-methoxy-2-methylphenyl)-3-[1-(pyrazin-2-yl)piperidin-3-yl]propanamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-(1H-imidazol-2-yl)benzamide
4-(4-methanesulfonylpiperazine-1-carbonyl)-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-4-(piperidin-1-yl)butanamide
N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
2-[({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)methyl]-3,4-dihydroquinazolin-4-one
[1-(4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenyl)ethyl]dimethylamine
(1S,5R)-3-{[4-(difluoromethoxy)phenyl]methyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
(5-{1-[(3-chloro-1H-indol-2-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
N-{[1-(4-chlorophenyl)cyclopropyl]methyl}-2-(pyrrolidin-3-yl)benzamide
3-methyl-5-(4-{2-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-imidazol-1-yl}phenyl)-4H-1,2,4-triazole
(1S,5R)-6-(cyclopropylmethyl)-3-[(3,5-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-2-(3-methoxyphenyl)ethan-1-one
1-(3,5-dimethoxybenzoyl)-4-(3-phenyl-1H-1,2,4-triazol-5-yl)piperidine
6-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-(2,6-dimethylpyridin-3-yl)-N-[4-(methylamino)butyl]pyrimidin-2-amine
2-(3-{2-amino-3-cyano-5H,6H,7H,8H,9H-cyclohepta[b]pyridin-4-yl}-1H-indol-1-yl)acetamide
2-(oxolan-2-ylmethyl)-9-(2-phenoxyacetyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-(3,4-difluorophenyl)piperidin-3-amine
N-[2-(1H-indol-1-yl)ethyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-butyl-2-[(dimethylcarbamoyl)amino]-N-(3-phenylprop-2-yn-1-yl)acetamide
3-[2-(3-aminoazetidin-1-yl)-2-oxoethyl]-3-benzyl-1-methyl-2,3-dihydro-1H-indol-2-one
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
5-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)pyrimidin-2-amine
3-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
(2S,4S)-4-[4-(dimethylamino)benzamido]-N-ethyl-1-(pent-2-yn-1-yl)pyrrolidine-2-carboxamide
4-[(4-fluorophenyl)methyl]-1-(1H-pyrrole-2-carbonyl)piperidine
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]cyclobutanecarboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[2-(morpholin-4-yl)butyl]-1,4-dithiepan-6-amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[1-(pyrimidin-4-yl)ethyl]benzamide
N-[(2-aminopyrimidin-5-yl)methyl]-2-(dimethylamino)-2-(3-fluorophenyl)-N-methylacetamide
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-[3-(4-fluorophenyl)propyl]piperidin-4-amine
N-[2-(2,3-dimethoxyphenyl)ethyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-methyl-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
4-cyclobutaneamido-N-(2-methoxyethyl)-N-(1-methylpiperidin-4-yl)benzamide
3-{2-amino-4-[3-(2-chlorophenyl)pyrrolidin-1-yl]-6-methylpyrimidin-5-yl}propanoic acid
5-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
(1R,5S,6R)-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
(3aS,6aS)-2-cyclopentyl-5-(2,4-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(4-methyl-5-{1-[(4-methylphenyl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
(1,4-dioxan-2-ylmethyl)(methyl){[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
3-{[(1-{thieno[3,2-d]pyrimidin-4-yl}piperidin-4-yl)amino]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-chloro-5-[3-hydroxy-3-(hydroxymethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
(2S,4S)-4-amino-N,N-diethyl-1-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]pyrrolidine-2-carboxamide