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N-[2-(adamantan-1-yl)-2-hydroxyethyl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-2-methyl-1-benzofuran-5-carboxamide
[(3S,5R)-1-(2,5-dimethylfuran-3-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
5-[(3S,5R)-3-(hydroxymethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidine-1-carbonyl]-1,2-oxazol-3-ol
(benzylsulfamoyl)[2-(4-fluorobenzenesulfonyl)ethyl]amine
N4-methyl-6-(propan-2-yloxy)-N4-[2-(1H-pyrazol-4-yl)ethyl]pyrimidine-2,4-diamine
N-[2-(azepan-1-yl)ethyl]-N-methylpyrazolo[1,5-a]pyridine-7-carboxamide
8-(5-chloro-2-methylbenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-phenyl-3-(piperidin-3-yl)-1-(quinolin-8-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(4-phenyl-5-{[1-(piperidin-3-yl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
1-methyl-4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
N-[4-(1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-imidazol-2-yl)phenyl]acetamide
(3S,4S)-1-[(4-methylphenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
4-{2-methyl-1-[4-(2-methylphenoxy)piperidin-1-yl]propan-2-yl}morpholine
3-(but-2-yn-1-yl)-5-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
3-(2-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-oxoethyl)-1,2,3-oxadiazol-3-ium-5-olate
N-methyl-6-oxo-1-(pyridin-2-ylmethyl)-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}piperidine-3-carboxamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-N-methylpiperidine-2-carboxamide
1-(4-ethylpiperazin-1-yl)-3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}propan-1-one
4-(1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine-4-carbonyl)morpholine
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(pyrrolidin-1-yl)propanamide
N-cyclopropyl-4-methoxy-3-({[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]carbamoyl}amino)benzamide
N-[3-(4-{[(1S)-1-carbamoyl-2-phenylethyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
4-[(furan-2-ylmethyl)amino]-N-(2-hydroxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(1S,5R)-3-benzyl-6-[(6-methylpyridin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(4-acetylphenoxy)-1-(2-benzylmorpholin-4-yl)ethan-1-one
2-{5-[2-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-methyl-1H-indole-6-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)(pyridin-3-ylmethyl)amine
4-(2-fluorobenzoyl)-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
2-ethyl-8-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
(2R,3S,6R)-3-(4-methylphenyl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
2-[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-[2-(1H-indol-3-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-(2-phenylethyl)-4-({1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}oxy)benzamide
5-(2-methoxy-4-methylphenoxymethyl)-N-[3-(propan-2-yloxy)propyl]-1,2-oxazole-3-carboxamide
3-(5-{[4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
1-(4,7-dimethylquinazolin-2-yl)-N-[1-(thiophen-2-yl)ethyl]azepan-4-amine
methyl 4-(5-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
(4aR,7aS)-1-ethyl-4-(6-hydroxyhexyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methoxy-1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[1-(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
4-(methoxymethyl)-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
1-ethyl-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
7-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]-4-methyl-1,2-dihydroquinolin-2-one
3-methyl-5-(2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(1,3-benzoxazol-2-yl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one