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8-acetyl-2-(1-phenylcyclopropanecarbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl[(2-methyl-1H-imidazol-4-yl)methyl](quinolin-8-ylmethyl)amine
(1R,5R)-6-[2-(2-fluorophenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
4-{[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}thiomorpholine
1-(oxan-4-yl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
2-(4-methoxy-3-methylphenyl)-N-methylbenzamide
methyl[(4-methyl-1H-imidazol-5-yl)methyl][1-(3-methylpyridin-2-yl)propan-2-yl]amine
1-(2-chlorophenyl)-3-{1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(3S,5S)-5-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-1-methylpyrrolidin-3-amine
1-{1-[2-(pyridin-2-yl)ethyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
1-methyl-3-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinoxalin-2-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl (2S)-1-({4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
3-methyl-1-(2-methylpropyl)-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazin-2-one
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(thiophen-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-{[5-(2-amino-6-methylpyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
1-(2-fluorophenyl)-4-[1-(furan-3-ylmethyl)piperidin-3-yl]piperazine
(1S,4S)-2-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
1-(2-methylphenyl)-3-(1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(1r,4r)-4-hydroxycyclohexyl]pyrimidine-5-carboxamide
7-(cyclobutylmethyl)-2-(2,2,3,3-tetramethylcyclopropanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-methanesulfonylethyl)-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
4-chloro-5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole
{imidazo[1,2-a]pyridin-3-ylmethyl}[(6-methoxy-2H-chromen-3-yl)methyl]methylamine
N-(1-{1-[3-(furan-2-yl)benzoyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
(3aS,6aS)-2-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(4-fluorophenyl)methyl]-4-(3-methoxypyrazin-2-yl)piperazin-2-one
1-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-3,3-diphenylpropan-1-one
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
[(2,3-difluoro-6-methoxyphenyl)methyl][2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
2-methoxy-N-{1-[1-(pyrrolidin-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(5-{1-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)methanol
N-(2-methylpropyl)-1-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yl)ethyl]amine
(1S,5R)-6-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-{[(4-methoxyphenyl)methyl]carbamoyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
1-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-methyl-3-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
methyl 4-{7-[(3,4-difluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-4-oxobutanoate
1-(4-{[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)-1H-1,2,4-triazole
2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
9-[2-hydroxy-4-(methylsulfanyl)butanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(4-chloro-2-methoxyphenoxymethyl)-N-(oxan-2-ylmethyl)-1,2-oxazole-3-carboxamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-[1-(2-methyl-1,3-benzothiazol-6-yl)-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl]acetamide
1-(4-ethylpiperazin-1-yl)-3-{1-[4-(4-hydroxyphenyl)butan-2-yl]piperidin-4-yl}propan-1-one
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine