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2-ethyl-6-methyl-4-oxo-N-(quinolin-3-ylmethyl)-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-ethyl-4-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazole
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)but-2-yn-1-one
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-(1H-pyrazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl 5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-(4-fluorophenyl)-N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
2-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)pyrrolidin-2-yl]-1,3-benzothiazole
2-(2H-1,3-benzodioxol-5-yl)-8-methyl-5-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
9-(3-hydroxy-4-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
8-cyclopentanecarbonyl-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
2-{2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamido}-N-methylacetamide
(3S,9aR)-8-(2,3-difluorobenzoyl)-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{1-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-methoxybenzamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-methylfuran-2-carboxamide
1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}-4-(pyridin-2-yl)piperidin-4-ol
N-{2-[1-(3-chloro-4-fluorobenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
N-cyclopropyl-1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
methyl 2-[4-(2-amino-6-tert-butyl-3-cyanopyridin-4-yl)-2-methoxyphenoxy]acetate
4-ethyl-3-({1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
1-{2-hydroxy-3-[2-methoxy-4-({[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amino}methyl)phenoxy]propyl}piperidin-4-ol
3-hydroxy-1-[(3-methylphenyl)methyl]-3-(morpholin-4-ylmethyl)piperidin-2-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
5-ethyl-N-[(1R)-1-(2-fluorophenyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
[1-({1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
3-fluoro-N-(1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)pyridin-3-ol
N-methyl-N-{3-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]propyl}aniline
11-methyl-5-(pyrimidin-4-ylmethyl)-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(methylsulfanyl)benzamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2,4-difluorophenyl)ethan-1-one
[(2,2-dimethyloxan-4-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
1,3-dimethyl-5-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)imidazolidine-2,4-dione
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[3-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
4-acetamido-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
1-[benzyl(methyl)amino]-3-[4-({[2-(propan-2-yloxy)ethyl]amino}methyl)phenoxy]propan-2-ol
methyl 6-(2-ethylbutyl)-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-{1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-5-methyl-1,2-oxazole
5-ethyl-N-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidin-2-amine
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(propan-2-yl)piperazin-1-yl]acetic acid
1-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{4-[2-(azocane-1-carbonyl)-4-methoxyphenoxy]piperidin-1-yl}ethan-1-one
3-[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-[(4-methylphenyl)methyl]propanamide
2-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyridine-3-carboxylic acid
2-(3-chloro-4-fluorophenoxy)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-(4-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
6-methyl-2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}pyridine-3-carboxylic acid