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N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[methyl(oxan-4-yl)amino]methyl}piperidin-2-one
N,N-dimethyl-4-(4-{[(2-methylphenyl)(pyridin-4-yl)methyl]amino}piperidin-1-yl)benzamide
N-(5-methyl-1,3-thiazol-2-yl)-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)benzamide
3-[2-(2-fluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
1-[5-(butan-2-yl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperidin-4-ol
3-benzyl-4-(2-methyl-1-benzofuran-5-carbonyl)piperazin-2-one
1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-3-ethylpiperidine-3-carboxylic acid
1-(1H-imidazol-2-ylmethyl)-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N,2-dimethyl-N-[2-(oxan-2-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[(5-fluoro-2-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(2,5-dioxo-1-propylimidazolidin-4-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-cyclopropyl-5-(1H-indole-2-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(azepane-1-carbonyl)-N-cyclopropyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-ethyl-5-[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(2-fluorophenyl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-5-(2,3,4-trimethoxyphenyl)benzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(methylamino)pyrimidin-2-yl]piperidin-3-ol
1-{[(3S)-3-ethylmorpholin-4-yl]sulfonyl}azepane
(4aS,8aR)-1-(2-aminoethyl)-6-(4-ethyl-5-methylthiophene-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
(2R,3R)-3-{[3-(azepan-1-yl)propyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-cyclohexyl-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
5-methoxy-3-methyl-2-{[3-(pyrimidin-4-yl)piperidin-1-yl]methyl}-1H-indole
N-({4-hydroxy-1-[(2-methyl-1-benzothiophen-3-yl)methyl]azepan-4-yl}methyl)cyclopropanecarboxamide
N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(6-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methanol
5-ethyl-N-(4,4,4-trifluorobutyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
methyl N-{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}carbamate
8-fluoro-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-2-carboxamide
[3-(2-phenoxyethyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]methanol
(2S,4R)-4-amino-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(pentylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-{[3-(2-hydroxyethyl)-4-(propan-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
(3R,4R)-4-(hydroxymethyl)-1-(4-methylpyridine-3-carbonyl)piperidin-3-ol
N,3-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-oxazole-5-carboxamide
ethyl 4-(2-phenoxyethyl)-1-(3-phenylprop-2-yn-1-yl)piperidine-4-carboxylate
N-[(2-fluorophenyl)methyl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
6-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methanol
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
3-({[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]carbamoyl}methyl)-1,2,3-oxadiazol-3-ium-5-olate
3-(2-methyl-1H-indol-1-yl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]propanamide
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-{[2-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
4-({1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
N-[4-methyl-3-({[2-(1,3-thiazol-4-yl)ethyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-[methyl(pyridin-3-ylmethyl)amino]acetamide