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3-cyclopropyl-1-methyl-4-[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N,N-dimethyl-2-{[2-(3-methylphenoxy)acetamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(4-fluorophenyl)-4-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]butan-1-one
2-(pyrrolidin-3-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}benzamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-(3-ethylphenyl)pyridine
1-[3-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidine-3-carboxamide
N-({1-[(2,6-difluoro-3-methylphenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}methyl)-2-methoxyacetamide
(3aS,7aR)-2-(3-cyclohexylpropanoyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-{[2-(propan-2-yloxy)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-(2-methoxyethyl)-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
(1R,7S)-6-(3-hydroxyazetidine-1-carbonyl)-3-[2-(4-methylphenyl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)amino)-1-phenylethan-1-ol
3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(2,5-dimethoxyphenyl)-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}acetamide
2-phenyl-4-[(2,3,4-trimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[6-(hydroxymethyl)pyridine-2-carbonyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
3-(2-ethylphenoxy)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}azetidine
2-(2-{4-phenyl-5-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}ethoxy)ethan-1-ol
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(thiophen-2-yl)butan-1-one
6-{[1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxy}pyridine-3-carboxylic acid
[(3-methoxyphenyl)methyl](methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
2-[5-(2,5-dihydro-1H-pyrrole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-methyl-1H-1,3-benzodiazole
N-(1-{7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
1-[2-(4-chlorophenyl)ethyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-(3-phenylcyclobutyl)-3-propoxypiperidine
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-methyl-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-{5-[1-(2,3-dimethylphenyl)piperidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)acetamide
1-[4-(dimethylamino)azepan-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]-5-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
5-methyl-1'-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-amino-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-4-carboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-N-[(3-methylphenyl)methyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
2-({cyclopropyl[(3-ethoxyphenyl)methyl]amino}methyl)-6-fluorophenol
8-(3-ethoxypropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
2-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}piperidine-3-carboxamide
methyl 3-benzamido-1-(furan-2-ylmethyl)-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol