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N-[4-(3-methoxyphenyl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-methyl-2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetamide
8-[3-(2-methylpropyl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]quinoline
(3R)-1-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}acetamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[4-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)carbamoyl}methoxy)phenyl]propanamide
2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
2-{4-[(2,3-dimethoxyphenyl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(3-phenylpropyl)-1,4-diazepane
methyl 8-(furan-2-ylmethyl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-[({imidazo[1,2-a]pyridin-3-ylmethyl}amino)methyl]piperidin-2-one
2-phenyl-5-(thiomorpholine-4-carbonyl)pyrimidin-4-ol
N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-4-(1H-pyrazol-4-yl)butanamide
(4aS,8aS)-2-(2-fluoro-4-methylbenzenesulfonyl)-decahydro-2,7-naphthyridin-4a-ol
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-[4-({3-hydroxy-1-[(3-methoxyphenyl)methyl]-2-oxopiperidin-3-yl}methyl)piperazin-1-yl]acetamide
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propan-2-ol
(1R,5S,8R)-3-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
4-[5-(3-chlorophenyl)furan-2-yl]-N-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
3-cyclohexyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-pyrazole-4-carboxamide
7-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-cyclopropanecarbonyl-1'-(4-methylpyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
5-(methoxymethyl)-N-methyl-N-(quinolin-6-ylmethyl)furan-2-carboxamide
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(2-methyl-1,3-thiazole-4-carbonyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}phenol
N-[3-({[2-(azepan-1-yl)ethyl](methyl)carbamoyl}amino)phenyl]butanamide
N-[2-(3-methylpyridin-2-yl)ethyl]-4-pentanamidobenzamide
N-[(3R,4S)-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
2-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-5-methoxypyridin-4-ol
6-methyl-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}imidazo[1,2-a]pyridine-2-carboxamide
2,3-dimethyl-5-phenyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-phenoxy-N-(pyridin-3-ylmethyl)acetamide
5-[1-(2,2-dimethylpropyl)pyrrolidin-2-yl]-N-(2,2,2-trifluoroethyl)thiophene-2-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-ethyl-4-methyl-6-[3-(pyridine-3-carbonyl)piperidin-1-yl]pyrimidine
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-[4-(pyrimidin-2-yloxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(2-chlorophenoxy)ethyl]-1-cyclopentyl-6-oxopiperidine-3-carboxamide
2-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-benzyl-N3-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-chlorophenyl)-N-(3-methoxypropyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
9-methyl-6-(1H-pyrazol-3-yl)-2,3,4,9-tetrahydro-1H-carbazol-1-one
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(1-methoxypropan-2-yl)-1,3-oxazole-4-carboxamide
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxypropan-1-one
1-benzyl-N,N-dimethyl-5-[(3-phenylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(methoxymethyl)-6-(piperidin-3-yl)-3,4-dihydropyrimidin-4-one
4-[(4-methylphenyl)methyl]-3-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one