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1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
(2S,4R)-4-amino-1-(4-acetamido-2-methylbenzoyl)-N-ethylpyrrolidine-2-carboxamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-3-(3-hydroxy-3-methylbutyl)benzamide
(4aR,8aS)-1-butyl-6-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
2-methoxy-1-(4-{[4-(methylsulfanyl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
3-[2-(2,6-difluorophenyl)ethyl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
N-methyl-4-(pyrrolidine-1-carbonyl)-6-(thiophen-3-ylmethyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
(1S,4S)-2-[5-(2-fluorophenyl)-1,2,4-triazin-3-yl]-2-azabicyclo[2.2.1]heptane
(2S)-3-(4-hydroxyphenyl)-2-{[4-(5-methylfuran-2-yl)phenyl]formamido}propanamide
(1S,5R)-3-(3,5-difluoropyridine-2-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
dimethyl({4-methyl-5-[1-(propane-2-sulfonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
2-(pyridin-2-yl)-5-{1-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-imidazol-2-yl}pyrimidine
3-(4-methylphenyl)-1-{4-[5-phenyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
(4S)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
4-[(4-methyl-5-{1-[2-(morpholin-4-yl)ethyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
[1-(2,3-dimethylquinoxaline-6-carbonyl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
1-{3-[(2S,6S)-6-butyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}propanamide
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-N-propylpyrimidin-2-amine
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-3-(3-hydroxy-1,2-oxazol-5-yl)propanamide
1-(2-methylphenyl)-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-1,4-diazepane
2-[1-(2-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
7-(5-chloropyridin-2-yl)-4-(1-methyl-1H-pyrrole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclohexyl-N-ethyl-5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carboxamide
N-[3-(1,3-benzothiazol-2-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5,6,7,8-tetrahydroquinoline
2-(7-methyl-1H-indol-3-yl)pyridine-3-carboxamide
7-(3-chlorophenyl)-4-(3-methylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-[2-(dimethylamino)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-({4-[5-(2-phenylacetamido)-1H-pyrazol-1-yl]piperidin-1-yl}methyl)benzoate
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{3',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]-5'-yl}ethan-1-one
2-(4-ethyl-2-methyl-1,3-thiazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(methylsulfanyl)-1-(4-phenyl-1,4-diazepan-1-yl)ethan-1-one
(2R,6R)-11-methoxy-4-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(1S,2S)-2-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)cyclohexan-1-ol
methyl 3-(2-methoxyacetamido)-5-[(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylformamido)methyl]benzoate
2-(5-fluoro-2-methylphenyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{1-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}ethan-1-one
N-cyclopentyl-N-[2-(dimethylamino)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
(3S,9aR)-3-(4-aminobutyl)-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-(propan-2-yl)pyridazin-3-amine
1-({5-[(3-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
4,6-dimethyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}pyrimidin-2-amine
2-(4-methylphenyl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]quinoline-4-carboxamide
3-hydroxy-3-[(4-methoxypiperidin-1-yl)methyl]-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
5-(2-chloro-4-fluorophenoxymethyl)-N-(1-phenylcyclopropyl)-1,2-oxazole-3-carboxamide
2-(4-chlorophenyl)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethan-1-one
4-hydroxy-1-[1-(1-phenylethyl)-1H-1,2,3,4-tetrazol-5-yl]piperidine-4-carboxylic acid
N-(2-methoxyethyl)-4-oxo-N-(thiophen-2-ylmethyl)-1,4-dihydroquinoline-2-carboxamide